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8FQ6

LBD of GluA2 flip Q isoform of AMPA receptor in complex with gain-of-function TARP gamma2, with 150mM CaCl2, 330uM CTZ, and 100mM L-glutamate (Open-Ca150)

Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1B, C, D, AGlutamate receptor 2polymer88999559.54UniProt (P19491)
Pfam (PF01094)
Pfam (PF10613)
Pfam (PF00060)
Pfam (PF00497)
In PDB
Rattus norvegicus (Norway rat)GluR-2,AMPA-selective glutamate receptor 2,GluR-B,GluR-K2,Glutamate receptor ionotropic,AMPA 2,GluA2
2B, C, D, AGLUTAMIC ACIDnon-polymer147.14Chemie (GLU)
3B, C, D, ACYCLOTHIAZIDEnon-polymer389.94Chemie (CYZ)
4waterwater18.016Chemie (HOH)
Sequence modifications
B, C, D, A: -20 - 868 (UniProt: P19491)
PDBExternal DatabaseDetails
Asp 848-insertion
Tyr 849-insertion
Lys 850-insertion
Asp 851-insertion
Asp 852-insertion
Asp 853-insertion
Asp 854Tyr 869conflict
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains4
Total formula weight398237.8
Non-Polymers*Number of molecules8
Total formula weight2148.0
All*Total formula weight400385.9
*Water molecules are not included.

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PDB entries from 2024-06-12

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