8F7S
Gi bound delta-opioid receptor in complex with deltorphin
Entity
Entity ID | Chain ID | Description | Type | Chain length | Formula weight | Number of molecules | DB Name (Accession) | Biological source | Descriptive keywords |
1 | R, D | Delta-type opioid receptor | polymer | 390 | 42651.0 | 2 | UniProt (P41143) Pfam (PF00001) In PDB | Homo sapiens (human) | D-OR-1,DOR-1 |
2 | P, Q | deltorphin | polymer | 8 | 781.9 | 2 | UniProt (P21850) In PDB | Phyllomedusa | [D-Ala2]-deltorphin II |
3 | A, F | Guanine nucleotide-binding protein G(i) subunit alpha-1 | polymer | 354 | 40445.1 | 2 | UniProt (P63096) Pfam (PF00503) In PDB | Homo sapiens (human) | Adenylate cyclase-inhibiting G alpha protein |
4 | B | Guanine nucleotide-binding protein G(I)/G(S)/G(T) subunit beta-1 | polymer | 353 | 39020.7 | 1 | UniProt (P54311) Pfam (PF00400) In PDB | Rattus norvegicus (Norway rat) | Transducin beta chain 1 |
5 | C | Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2 | polymer | 68 | 7563.8 | 1 | UniProt (P63212) Pfam (PF00631) In PDB | Bos taurus (cattle) | G gamma-I |
6 | R, D | CHOLESTEROL | non-polymer | 386.7 | 5 | Chemie (CLR) | |||
7 | R, D | PALMITIC ACID | non-polymer | 256.4 | 12 | Chemie (PLM) |
Sequence modifications
R, D: 2 - 372 (UniProt: P41143)
P, Q: 1 - 7 (UniProt: P21850)
A, F: 1 - 354 (UniProt: P63096)
B: 7 - 345 (UniProt: P54311)
PDB | External Database | Details |
---|---|---|
Asp -9 | - | expression tag |
Tyr -8 | - | expression tag |
Lys -7 | - | expression tag |
Asp -6 | - | expression tag |
Asp -5 | - | expression tag |
Asp -4 | - | expression tag |
Asp -3 | - | expression tag |
Val -2 | - | expression tag |
Asp -1 | - | expression tag |
Ala 0 | - | expression tag |
Ser 1 | - | expression tag |
Val 73 | Gly 73 | conflict |
Ser 90 | Asn 90 | conflict |
Gly 95 | Asp 95 | conflict |
Ser 131 | Asn 131 | conflict |
Cys 143 | Ser 143 | conflict |
Val 268 | Gly 268 | conflict |
Ile 309 | Ala 309 | conflict |
His 373 | - | expression tag |
His 374 | - | expression tag |
His 375 | - | expression tag |
His 376 | - | expression tag |
His 377 | - | expression tag |
His 378 | - | expression tag |
His 379 | - | expression tag |
His 380 | - | expression tag |
PDB | External Database | Details |
---|---|---|
Dal 2 | Ala 108 | variant |
Nh2 8 | - | amidation |
PDB | External Database | Details |
---|---|---|
Ala 203 | Gly 203 | conflict |
Ser 326 | Ala 326 | conflict |
PDB | External Database | Details |
---|---|---|
Met -7 | - | expression tag |
His -6 | - | expression tag |
His -5 | - | expression tag |
His -4 | - | expression tag |
His -3 | - | expression tag |
His -2 | - | expression tag |
His -1 | - | expression tag |
His 0 | - | expression tag |
His 1 | - | expression tag |
Gly 2 | - | expression tag |
Ser 3 | - | expression tag |
Leu 4 | - | expression tag |
Leu 5 | - | expression tag |
Gln 6 | - | expression tag |
Sequence viewer
Contents of the asymmetric unit
Polymers | Number of chains | 8 |
Total formula weight | 214340.3 | |
Non-Polymers* | Number of molecules | 17 |
Total formula weight | 5010.4 | |
All* | Total formula weight | 219350.7 |