7XAV
Structure of somatostatin receptor 2 bound with lanreotide.
Entity
Entity ID | Chain ID | Description | Type | Chain length | Formula weight | Number of molecules | DB Name (Accession) | Biological source | Descriptive keywords |
1 | A | Somatostatin receptor type 2,LargeBit | polymer | 563 | 63274.4 | 1 | UniProt (P30874) Pfam (PF00001) In PDB | Homo sapiens (human) | SS-2-R,SS2-R,SS2R,SRIF-1 |
2 | B | Guanine nucleotide-binding protein G(i) subunit alpha-1 | polymer | 354 | 40472.1 | 1 | UniProt (P63096) Pfam (PF00503) In PDB | Homo sapiens (human) | Adenylate cyclase-inhibiting G alpha protein |
3 | C | Guanine nucleotide-binding protein G(I)/G(S)/G(T) subunit beta-1 | polymer | 354 | 38975.6 | 1 | UniProt (P62871) Pfam (PF00400) In PDB | Bos taurus (cattle) | Transducin beta chain 1 |
4 | D | Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2 | polymer | 71 | 7861.1 | 1 | UniProt (P63212) Pfam (PF00631) In PDB | Bos taurus (cattle) | G gamma-I |
5 | E | ScFv16 | polymer | 304 | 32768.5 | 1 | Rattus | ||
6 | F | Lanreotide | polymer | 9 | 1098.3 | 1 | synthetic construct |
Sequence modifications
A: 1 - 359 (UniProt: P30874)
A: 360 - 517 (PDB: 7XAV)
B: 1 - 354 (UniProt: P63096)
C: 2 - 340 (UniProt: P62871)
PDB | External Database | Details |
---|---|---|
Met -45 | - | initiating methionine |
Lys -44 | - | expression tag |
Thr -43 | - | expression tag |
Ile -42 | - | expression tag |
Ile -41 | - | expression tag |
Ala -40 | - | expression tag |
Leu -39 | - | expression tag |
Ser -38 | - | expression tag |
Tyr -37 | - | expression tag |
Ile -36 | - | expression tag |
Phe -35 | - | expression tag |
Cys -34 | - | expression tag |
Leu -33 | - | expression tag |
Val -32 | - | expression tag |
Phe -31 | - | expression tag |
Ala -30 | - | expression tag |
Asp -29 | - | expression tag |
Tyr -28 | - | expression tag |
Lys -27 | - | expression tag |
Asp -26 | - | expression tag |
Asp -25 | - | expression tag |
Asp -24 | - | expression tag |
Asp -23 | - | expression tag |
Lys -22 | - | expression tag |
Gly -21 | - | expression tag |
Ser -20 | - | expression tag |
Gly -19 | - | expression tag |
Ser -18 | - | expression tag |
His -17 | - | expression tag |
His -16 | - | expression tag |
His -15 | - | expression tag |
His -14 | - | expression tag |
His -13 | - | expression tag |
His -12 | - | expression tag |
His -11 | - | expression tag |
His -10 | - | expression tag |
His -9 | - | expression tag |
His -8 | - | expression tag |
Leu -7 | - | expression tag |
Glu -6 | - | expression tag |
Val -5 | - | expression tag |
Leu -4 | - | expression tag |
Phe -3 | - | expression tag |
Gln -2 | - | expression tag |
Gly -1 | - | expression tag |
Pro 0 | - | expression tag |
B: 1 - 354 (UniProt: P63096)
PDB | External Database | Details |
---|---|---|
Asn 47 | Ser 47 | conflict |
Ala 203 | Gly 203 | conflict |
Ser 326 | Ala 326 | conflict |
PDB | External Database | Details |
---|---|---|
Met -10 | - | initiating methionine |
His -9 | - | expression tag |
His -8 | - | expression tag |
His -7 | - | expression tag |
His -6 | - | expression tag |
His -5 | - | expression tag |
His -4 | - | expression tag |
Gly -3 | - | expression tag |
Ser -2 | - | expression tag |
Leu -1 | - | expression tag |
Leu 0 | - | expression tag |
Gln 1 | - | expression tag |
Gly 341 | - | expression tag |
Ser 342 | - | expression tag |
Ser 343 | - | expression tag |
Sequence viewer
Contents of the asymmetric unit
Polymers | Number of chains | 6 |
Total formula weight | 184450.0 | |
All* | Total formula weight | 184450.0 |