7VKO
Crystal structure of TrkA kinase with repotrectinib
Entity
Entity ID | Chain ID | Description | Type | Chain length | Formula weight | Number of molecules | DB Name (Accession) | Biological source | Descriptive keywords |
1 | A | Tyrosine-protein kinase receptor | polymer | 326 | 37235.8 | 1 | UniProt (J3KP20) Pfam (PF07714) UniProt (by SIFTS) (P04629) In PDB | Homo sapiens (Human) | |
2 | A | Repotrectinib | non-polymer | 355.4 | 1 | Chemie (7GI) | |||
3 | A | SULFATE ION | non-polymer | 96.1 | 5 | Chemie (SO4) | |||
4 | water | water | 18.0 | 21 | Chemie (HOH) |
Sequence modifications
A: 502 - 796 (UniProt: J3KP20)
PDB | External Database | Details |
---|---|---|
Met 471 | - | initiating methionine |
Ser 472 | - | expression tag |
Tyr 473 | - | expression tag |
Tyr 474 | - | expression tag |
His 475 | - | expression tag |
His 476 | - | expression tag |
His 477 | - | expression tag |
His 478 | - | expression tag |
His 479 | - | expression tag |
His 480 | - | expression tag |
Asp 481 | - | expression tag |
Tyr 482 | - | expression tag |
Asp 483 | - | expression tag |
Ile 484 | - | expression tag |
Pro 485 | - | expression tag |
Thr 486 | - | expression tag |
Thr 487 | - | expression tag |
Glu 488 | - | expression tag |
Asn 489 | - | expression tag |
Leu 490 | - | expression tag |
Tyr 491 | - | expression tag |
Phe 492 | - | expression tag |
Gln 493 | - | expression tag |
Gly 494 | - | expression tag |
Ala 495 | - | expression tag |
Met 496 | - | expression tag |
Gly 497 | - | expression tag |
Ser 498 | - | expression tag |
Gly 499 | - | expression tag |
Ile 500 | - | expression tag |
Arg 501 | - | expression tag |
Sequence viewer
Contents of the asymmetric unit
Polymers | Number of chains | 1 |
Total formula weight | 37235.8 | |
Non-Polymers* | Number of molecules | 6 |
Total formula weight | 835.7 | |
All* | Total formula weight | 38071.5 |