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7OIS

mPI3Kd in complex with compound 7

This is a non-PDB format compatible entry.
Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1AAAPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoformpolymer1084124834.51UniProt (O35904)
Pfam (PF02192)
Pfam (PF00794)
Pfam (PF00792)
Pfam (PF00613)
Pfam (PF00454)
In PDB
Mus musculus (Mouse)PI3-kinase subunit delta,PI3K-delta,PI3Kdelta,PtdIns-3-kinase subunit delta,Phosphatidylinositol 4,5-bisphosphate 3-kinase 110 kDa catalytic subunit delta,PtdIns-3-kinase subunit p110-delta,p110delta
2AAASODIUM IONnon-polymer23.01Chemie (NA)
3AAAN-[5-[2-[(1S)-1-cyclopropylethyl]-7-[(3-methylsulfonylphenyl)sulfamoyl]-1-oxidanylidene-3H-isoindol-5-yl]-4-methyl-1,3-thiazol-2-yl]ethanamidenon-polymer588.71Chemie (VEW)
4waterwater18.01532Chemie (HOH)
Sequence modifications
AAA: -6 - 1044 (UniProt: O35904)
PDBExternal DatabaseDetails
Met -39-initiating methionine
Ser -38-expression tag
Tyr -37-expression tag
His -36-expression tag
Asn -35-expression tag
His -34-expression tag
Asn -33-expression tag
His -32-expression tag
Asn -31-expression tag
His -30-expression tag
Asn -29-expression tag
His -28-expression tag
Asn -27-expression tag
His -26-expression tag
Asn -25-expression tag
Asp -24-expression tag
Tyr -23-expression tag
Asp -22-expression tag
Ile -21-expression tag
Pro -20-expression tag
Thr -19-expression tag
Thr -18-expression tag
Glu -17-expression tag
Asn -16-expression tag
Leu -15-expression tag
Tyr -14-expression tag
Phe -13-expression tag
Gln -12-expression tag
Gly -11-expression tag
Ala -10-expression tag
Met -9-expression tag
Asp -8-expression tag
Leu -7-expression tag
Glu 99-insertion
Asn 100-insertion
Leu 101-insertion
Tyr 102-insertion
Phe 103-insertion
Gln 104-insertion
Gly 105-insertion
Gln 510-insertion
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains1
Total formula weight124834.5
Non-Polymers*Number of molecules2
Total formula weight611.7
All*Total formula weight125446.2
*Water molecules are not included.

221051

PDB entries from 2024-06-12

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