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6VNK

JAK2 JH1 in complex with PN4-073

Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1D, B, C, ATyrosine-protein kinase JAK2polymer30836455.44UniProt (O60674)
Pfam (PF07714)
In PDB
Homo sapiens (Human)Janus kinase 2,JAK-2
2D, B, C, A(3R)-3-cyclopentyl-3-[4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl]propanenitrilenon-polymer306.44Chemie (RXT)
3waterwater18.0462Chemie (HOH)
Sequence modifications
D, B, C, A: 840 - 1132 (UniProt: O60674)
PDBExternal DatabaseDetails
His 825-expression tag
His 826-expression tag
His 827-expression tag
His 828-expression tag
His 829-expression tag
His 830-expression tag
His 831-expression tag
His 832-expression tag
Glu 833-expression tag
Asn 834-expression tag
Leu 835-expression tag
Tyr 836-expression tag
Phe 837-expression tag
Gln 838-expression tag
Gly 839-expression tag
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains4
Total formula weight145821.8
Non-Polymers*Number of molecules4
Total formula weight1225.5
All*Total formula weight147047.2
*Water molecules are not included.

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PDB entries from 2024-06-12

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