6GG8
Mineralocorticoid receptor in complex with (s)-13
Entity
Entity ID | Chain ID | Description | Type | Chain length | Formula weight | Number of molecules | DB Name (Accession) | Biological source | Descriptive keywords |
1 | A | Mineralocorticoid receptor | polymer | 305 | 34806.7 | 1 | UniProt (P08235) Pfam (PF00104) In PDB | Homo sapiens (Human) | MR,Nuclear receptor subfamily 3 group C member 2 |
2 | B | Nuclear receptor coactivator 1 | polymer | 15 | 1726.0 | 1 | UniProt (Q15788) In PDB | Homo sapiens (Human) | NCoA-1,Class E basic helix-loop-helix protein 74,bHLHe74,Protein Hin-2,RIP160,Renal carcinoma antigen NY-REN-52,Steroid receptor coactivator 1,SRC-1 |
3 | A | (4S)-2-METHYL-2,4-PENTANEDIOL | non-polymer | 118.2 | 1 | Chemie (MPD) | |||
4 | A | [(3~{R})-7-fluoranyl-4-[(3-oxidanylidene-4~{H}-1,4-benzoxazin-6-yl)carbonyl]-2,3-dihydro-1,4-benzoxazin-3-yl]methanesulfonamide | non-polymer | 421.4 | 1 | Chemie (EY8) | |||
5 | water | water | 18.0 | 186 | Chemie (HOH) |
Sequence modifications
A: 735 - 984 (UniProt: P08235)
PDB | External Database | Details |
---|---|---|
Met 713 | - | initiating methionine |
His 714 | - | expression tag |
Asn 715 | - | expression tag |
His 716 | - | expression tag |
Asn 717 | - | expression tag |
His 718 | - | expression tag |
Asn 719 | - | expression tag |
His 720 | - | expression tag |
Asn 721 | - | expression tag |
His 722 | - | expression tag |
Asn 723 | - | expression tag |
His 724 | - | expression tag |
Asn 725 | - | expression tag |
Gly 726 | - | expression tag |
Gly 727 | - | expression tag |
Glu 728 | - | expression tag |
Asn 729 | - | expression tag |
Leu 730 | - | expression tag |
Tyr 731 | - | expression tag |
Phe 732 | - | expression tag |
Gln 733 | - | expression tag |
Gly 734 | - | expression tag |
Ser 808 | Cys 808 | conflict |
Ser 910 | Cys 910 | conflict |
Gly 985 | - | expression tag |
Gly 986 | - | expression tag |
Ser 987 | - | expression tag |
Leu 988 | - | expression tag |
Val 989 | - | expression tag |
Pro 990 | - | expression tag |
Arg 991 | - | expression tag |
Gly 992 | - | expression tag |
Ser 993 | - | expression tag |
Gly 994 | - | expression tag |
Gly 995 | - | expression tag |
Gly 996 | - | expression tag |
Ser 997 | - | expression tag |
Gly 998 | - | expression tag |
Gly 999 | - | expression tag |
Ser 1000 | - | expression tag |
Gly 1001 | - | expression tag |
Gly 1002 | - | expression tag |
Pro 1003 | - | expression tag |
Gln 1004 | - | expression tag |
Ala 1005 | - | expression tag |
Gln 1006 | - | expression tag |
Gln 1007 | - | expression tag |
Lys 1008 | - | expression tag |
Ser 1009 | - | expression tag |
Leu 1010 | - | expression tag |
Leu 1011 | - | expression tag |
Gln 1012 | - | expression tag |
Gln 1013 | - | expression tag |
Leu 1014 | - | expression tag |
Leu 1015 | - | expression tag |
Thr 1016 | - | expression tag |
Glu 1017 | - | expression tag |
Sequence viewer
Contents of the asymmetric unit
Polymers | Number of chains | 2 |
Total formula weight | 36532.6 | |
Non-Polymers* | Number of molecules | 2 |
Total formula weight | 539.6 | |
All* | Total formula weight | 37072.2 |