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6DQC

LINKED KDM5A JMJ DOMAIN BOUND TO THE INHIBITOR N50 i.e. 2-(4-((2-(dimethylamino)ethyl)(ethyl)carbamoyl)-5-(4-methoxyphenyl)-1H-pyrazol-1-yl)isonicotinic acid

Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1ALinked KDM5A Jmj Domainpolymer33037944.81UniProt (P29375)
Pfam (PF02375)
Pfam (PF02373)
In PDB
Homo sapiens (Human)Histone demethylase JARID1A,Jumonji/ARID domain-containing protein 1A,Retinoblastoma-binding protein 2,RBBP-2,Histone demethylase JARID1A,Jumonji/ARID domain-containing protein 1A,Retinoblastoma-binding protein 2,RBBP-2
2A2-[4-{[2-(dimethylamino)ethyl](ethyl)carbamoyl}-5-(4-methoxyphenyl)-1H-pyrazol-1-yl]pyridine-4-carboxylic acidnon-polymer437.51Chemie (H5Y)
3AMANGANESE (II) IONnon-polymer54.91Chemie (MN)
4ADIMETHYL SULFOXIDEnon-polymer78.11Chemie (DMS)
5AGLYCEROLnon-polymer92.11Chemie (GOL)
6ASULFATE IONnon-polymer96.11Chemie (SO4)
7waterwater18.0162Chemie (HOH)
Sequence modifications
A: 1 - 87 (UniProt: P29375)
PDBExternal DatabaseDetails
His -1-expression tag
Asn 0-expression tag
A: 348 - 588 (UniProt: P29375)
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains1
Total formula weight37944.8
Non-Polymers*Number of molecules5
Total formula weight758.7
All*Total formula weight38703.6
*Water molecules are not included.

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PDB entries from 2024-08-14

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