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5VED

PAK4 kinase domain in complex with Staurosporine

Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1A
(A)
Serine/threonine-protein kinase PAK 4polymer31936025.71UniProt (O96013)
Pfam (PF00069)
Homo sapiens (Human)p21-activated kinase 4,PAK-4
2B
(A)
STAUROSPORINEnon-polymer466.51Chemie (STU)
PubChem (5279)
PubChem (44259)
PubChem (71203703)
PubChem (42610657)
PubChem (44299148)
PubChem (25322871)
PubChem (28684983)
PubChem (451705)
PubChem (44120114)
PubChem (44537813)
PubChem (49831000)
PubChem (46864193)
PubChem (68262703)
PubChem (68306294)
PubChem (5459111)
PubChem (73953205)
PubChem (6419748)
PubChem (86306248)
PubChem (358479)
PubChem (9804568)
PubChem (9937179)
PubChem (5280487)
PubChem (5311103)
PubChem (6711321)
PubChem (9956178)
PubChem (122130844)
PubChem (12046017)
PubChem (143163481)
PubChem (143224059)
PubChem (143494026)
PubChem (162978898)
3C
(A)
waterwater18.015Chemie (HOH)
Sequence modifications
A: 286 - 591 (UniProt: O96013)
PDBExternal DatabaseDetails
Gly 273-expression tag
Ala 274-expression tag
Arg 275-expression tag
Ala 276-expression tag
Arg 277-expression tag
Gln 278-expression tag
Glu 279-expression tag
Asn 280-expression tag
Gly 281-expression tag
Met 282-expression tag
Pro 283-expression tag
Glu 284-expression tag
Lys 285-expression tag
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains1
Total formula weight36025.7
Non-Polymers*Number of molecules1
Total formula weight466.5
All*Total formula weight36492.3
*Water molecules are not included.

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PDB entries from 2026-04-01

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