5UFI
DCN1 bound to DI-591
Entity
Entity ID | Chain ID | Description | Type | Chain length | Formula weight | Number of molecules | DB Name (Accession) | Biological source | Descriptive keywords |
1 | A, B, C, D | DCN1-like protein 1 | polymer | 225 | 26251.9 | 4 | UniProt (Q96GG9) Pfam (PF03556) In PDB | Homo sapiens (Human) | DCUN1 domain-containing protein 1,Defective in cullin neddylation protein 1-like protein 1,Squamous cell carcinoma-related oncogene |
2 | A, B, C, D | N-[(1S)-1-cyclohexyl-2-{[3-(morpholin-4-yl)propanoyl]amino}ethyl]-N~2~-propanoyl-3-[6-(propan-2-yl)-1,3-benzothiazol-2-yl]-L-alaninamide | non-polymer | 585.8 | 4 | BIRD (PRD_002263) Chemie (8B1) | |||
3 | water | water | 18.0 | 40 | Chemie (HOH) |
Sequence modifications
A, B, C, D: 58 - 259 (UniProt: Q96GG9)
PDB | External Database | Details |
---|---|---|
Met 35 | - | initiating methionine |
Ser 36 | - | expression tag |
Tyr 37 | - | expression tag |
Tyr 38 | - | expression tag |
His 39 | - | expression tag |
His 40 | - | expression tag |
His 41 | - | expression tag |
His 42 | - | expression tag |
His 43 | - | expression tag |
His 44 | - | expression tag |
Leu 45 | - | expression tag |
Glu 46 | - | expression tag |
Ser 47 | - | expression tag |
Thr 48 | - | expression tag |
Ser 49 | - | expression tag |
Leu 50 | - | expression tag |
Tyr 51 | - | expression tag |
Lys 52 | - | expression tag |
Lys 53 | - | expression tag |
Ala 54 | - | expression tag |
Gly 55 | - | expression tag |
Thr 56 | - | expression tag |
Met 57 | - | expression tag |
Sequence viewer
Contents of the asymmetric unit
Polymers | Number of chains | 4 |
Total formula weight | 105007.5 | |
Non-Polymers* | Number of molecules | 4 |
Total formula weight | 2343.2 | |
All* | Total formula weight | 107350.7 |