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5TF5

CRYSTAL STRUCTURE OF HUMAN KAT-2 IN COMPLEX WITH A REVERSIBLE INHIBITOR

Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1A, B
(A, B)
Kynurenine/alpha-aminoadipate aminotransferase, mitochondrialpolymer42547628.62UniProt (Q8N5Z0)
Pfam (PF00155)
Homo sapiens (Human)KAT/AadAT,2-aminoadipate aminotransferase,2-aminoadipate transaminase,Alpha-aminoadipate aminotransferase,AadAT,Kynurenine aminotransferase II,Kynurenine--oxoglutarate aminotransferase II,Kynurenine--oxoglutarate transaminase 2,Kynurenine--oxoglutarate transaminase II
2C
(B)
(2R)-2-(5,6-dichloro-1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)-3-phenylpropanoic acidnon-polymer364.21Chemie (7AR)
3D, E
(A, B)
waterwater18.0682Chemie (HOH)
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains2
Total formula weight95257.1
Non-Polymers*Number of molecules1
Total formula weight364.2
All*Total formula weight95621.3
*Water molecules are not included.

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PDB entries from 2025-12-24

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