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5T8F

p110delta/p85alpha with taselisib (GDC-0032)

Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1APhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoformpolymer1015116187.21UniProt (O00329)
Pfam (PF02192)
Pfam (PF00794)
Pfam (PF00792)
Pfam (PF00613)
Pfam (PF00454)
In PDB
Homo sapiens (Human)PtdIns-3-kinase subunit delta,Phosphatidylinositol 4,5-bisphosphate 3-kinase 110 kDa catalytic subunit delta,p110delta
2BPhosphatidylinositol 3-kinase regulatory subunit alphapolymer16920879.61UniProt (P23727)
Pfam (PF16454)
In PDB
Bos taurus (Bovine)PtdIns-3-kinase regulatory subunit alpha,Phosphatidylinositol 3-kinase 85 kDa regulatory subunit alpha,PtdIns-3-kinase regulatory subunit p85-alpha
3A2-methyl-2-(4-{2-[3-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-5-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-1H-pyrazol-1-yl)propanamidenon-polymer460.51Chemie (799)
4waterwater18.01Chemie (HOH)
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains2
Total formula weight137066.7
Non-Polymers*Number of molecules1
Total formula weight460.5
All*Total formula weight137527.3
*Water molecules are not included.

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PDB entries from 2024-07-10

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