5NG5
multi-drug efflux; membrane transport; RND superfamily; Drug resistance
Entity
Entity ID | Chain ID | Description | Type | Chain length | Formula weight | Number of molecules | DB Name (Accession) | Biological source | Descriptive keywords |
1 | E, D, G, H, A... | Multidrug efflux pump subunit AcrA | polymer | 373 | 39800.7 | 6 | UniProt (P0AE06) Pfam (PF00529) Pfam (PF16576) In PDB | Escherichia coli | AcrAB-TolC multidrug efflux pump subunit AcrA,Acridine resistance protein A |
2 | F, I, C | Outer membrane protein TolC | polymer | 493 | 53783.4 | 3 | UniProt (P02930) Pfam (PF02321) In PDB | Escherichia coli | Multidrug efflux pump subunit TolC,Outer membrane factor TolC |
3 | K, L, J | Multidrug efflux pump subunit AcrB | polymer | 1049 | 113665.2 | 3 | UniProt (P31224) Pfam (PF00873) In PDB | Escherichia coli | AcrAB-TolC multidrug efflux pump subunit AcrB,Acridine resistance protein B |
4 | M, N, O | Multidrug efflux pump accessory protein AcrZ | polymer | 54 | 5995.2 | 3 | UniProt (P0AAW9) Pfam (PF10766) In PDB | Escherichia coli | AcrAB-TolC multidrug efflux pump accessory protein AcrZ,Acridine resistance protein Z |
5 | K, L, J | 6-[2-(3,4-dimethoxyphenyl)ethylsulfanyl]-8-[4-(2-methoxyethyl)piperazin-1-yl]-3,3-dimethyl-1,4-dihydropyrano[3,4-c]pyridine-5-carbonitrile | non-polymer | 526.7 | 3 | Chemie (5QF) |
Sequence modifications
E, D, G, H, A, B: 25 - 397 (UniProt: P0AE06)
M, N, O: 1 - 49 (UniProt: P0AAW9)
PDB | External Database | Details |
---|---|---|
Met 223 | Phe 223 | conflict |
Met 224 | Leu 224 | conflict |
Met 287 | Leu 287 | conflict |
Met 288 | Leu 288 | conflict |
PDB | External Database | Details |
---|---|---|
His 50 | - | expression tag |
His 51 | - | expression tag |
His 52 | - | expression tag |
His 53 | - | expression tag |
His 54 | - | expression tag |
Sequence viewer
Contents of the asymmetric unit
Polymers | Number of chains | 15 |
Total formula weight | 759135.0 | |
Non-Polymers* | Number of molecules | 3 |
Total formula weight | 1580.1 | |
All* | Total formula weight | 760715.1 |