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5L2T

The X-ray co-crystal structure of human CDK6 and Ribociclib.

Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1A
(A)
Cyclin-dependent kinase 6polymer30735019.21UniProt (Q00534)
Pfam (PF00069)
Homo sapiens (Human)Cell division protein kinase 6,Serine/threonine-protein kinase PLSTIRE
2B
(A)
7-cyclopentyl-N,N-dimethyl-2-{[5-(piperazin-1-yl)pyridin-2-yl]amino}-7H-pyrrolo[2,3-d]pyrimidine-6-carboxamidenon-polymer434.51Chemie (6ZZ)
3C
(A)
waterwater18.02Chemie (HOH)
Sequence modifications
A: 1 - 301 (UniProt: Q00534)
PDBExternal DatabaseDetails
His 302-expression tag
His 303-expression tag
His 304-expression tag
His 305-expression tag
His 306-expression tag
His 307-expression tag
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains1
Total formula weight35019.2
Non-Polymers*Number of molecules1
Total formula weight434.5
All*Total formula weight35453.8
*Water molecules are not included.

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PDB entries from 2025-07-30

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