5L1H
AMPA subtype ionotropic glutamate receptor GluA2 in complex with noncompetitive inhibitor GYKI53655
Entity
Entity ID | Chain ID | Description | Type | Chain length | Formula weight | Number of molecules | DB Name (Accession) | Biological source | Descriptive keywords |
1 | A, B, C, D | Glutamate receptor 2 | polymer | 803 | 89805.7 | 4 | UniProt (P19491) Pfam (PF01094) Pfam (PF10613) Pfam (PF00060) In PDB | Rattus norvegicus (Rat) | GluR-2,AMPA-selective glutamate receptor 2,GluR-B,GluR-K2,Glutamate receptor ionotropic,AMPA 2,GluA2 |
2 | A, B, C, D | 2-acetamido-2-deoxy-beta-D-glucopyranose | non-polymer | 221.2 | 4 | Chemie (NAG) | |||
3 | A, B, C, D | (8R)-5-(4-aminophenyl)-N,8-dimethyl-8,9-dihydro-2H,7H-[1,3]dioxolo[4,5-h][2,3]benzodiazepine-7-carboxamide | non-polymer | 352.4 | 4 | Chemie (GYK) |
Sequence modifications
A, B, C, D: 10 - 544 (UniProt: P19491)
A, B, C, D: 567 - 826 (UniProt: P19491)
PDB | External Database | Details |
---|---|---|
Glu 241 | Asn 256 | engineered mutation |
- | Val 397 | deletion |
- | Thr 398 | deletion |
- | Leu 402 | deletion |
- | Pro 403 | deletion |
- | Ser 404 | deletion |
- | Gly 405 | deletion |
Asp 385 | Asn 406 | engineered mutation |
Gln 392 | Asn 413 | engineered mutation |
PDB | External Database | Details |
---|---|---|
Asp 564 | - | linker |
Thr 565 | - | linker |
Asp 566 | - | linker |
Ala 589 | Cys 610 | engineered mutation |
Gly 827 | - | cloning artifact |
Leu 828 | - | cloning artifact |
Val 829 | - | cloning artifact |
Pro 830 | - | cloning artifact |
Arg 831 | - | cloning artifact |
Sequence viewer
Contents of the asymmetric unit
Polymers | Number of chains | 4 |
Total formula weight | 359222.9 | |
Non-Polymers* | Number of molecules | 8 |
Total formula weight | 2294.4 | |
All* | Total formula weight | 361517.3 |