5JFS
Crystal structure of TrkA in complex with PF-00593174
Entity
Entity ID | Chain ID | Description | Type | Chain length | Formula weight | Number of molecules | DB Name (Accession) | Biological source | Descriptive keywords |
1 | A | High affinity nerve growth factor receptor | polymer | 308 | 35101.6 | 1 | UniProt (P04629) Pfam (PF07714) In PDB | Homo sapiens (Human) | Neurotrophic tyrosine kinase receptor type 1,TRK1-transforming tyrosine kinase protein,Tropomyosin-related kinase A,Tyrosine kinase receptor A,Trk-A,gp140trk,p140-TrkA |
2 | A | N-{4-[4-amino-7-(propan-2-yl)-7H-pyrrolo[2,3-d]pyrimidine-5-carbonyl]pyridin-2-yl}-N'-(2,4-difluorophenyl)urea | non-polymer | 451.4 | 1 | Chemie (6K0) | |||
3 | water | water | 18.0 | 364 | Chemie (HOH) |
Sequence modifications
A: 502 - 796 (UniProt: P04629)
PDB | External Database | Details |
---|---|---|
Met 489 | - | initiating methionine |
His 490 | - | expression tag |
His 491 | - | expression tag |
His 492 | - | expression tag |
His 493 | - | expression tag |
His 494 | - | expression tag |
His 495 | - | expression tag |
Leu 496 | - | expression tag |
Val 497 | - | expression tag |
Pro 498 | - | expression tag |
Arg 499 | - | expression tag |
Gly 500 | - | expression tag |
Ser 501 | - | expression tag |
Sequence viewer
Contents of the asymmetric unit
Polymers | Number of chains | 1 |
Total formula weight | 35101.6 | |
Non-Polymers* | Number of molecules | 1 |
Total formula weight | 451.4 | |
All* | Total formula weight | 35553.0 |