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4YZC

Crystal structure of pIRE1alpha in complex with staurosporine

Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1A, B
(A, B)
Serine/threonine-protein kinase/endoribonuclease IRE1polymer40546850.52UniProt (O75460)
Pfam (PF00069)
Pfam (PF06479)
Homo sapiens (Human)Endoplasmic reticulum-to-nucleus signaling 1,Inositol-requiring protein 1,hIRE1p,Ire1-alpha,IRE1a
2C, D
(A, B)
STAUROSPORINEnon-polymer466.52Chemie (STU)
PubChem (5279)
PubChem (44259)
PubChem (451705)
PubChem (5459111)
PubChem (6419748)
PubChem (9804568)
PubChem (9937179)
PubChem (71203703)
PubChem (42610657)
PubChem (44299148)
PubChem (25322871)
PubChem (28684983)
PubChem (49831000)
PubChem (44120114)
PubChem (44537813)
PubChem (46864193)
PubChem (358479)
PubChem (5280487)
PubChem (5311103)
PubChem (6711321)
PubChem (9956178)
PubChem (12046017)
PubChem (68262703)
PubChem (68306294)
PubChem (73953205)
PubChem (86306248)
PubChem (122130844)
PubChem (143163481)
PubChem (143224059)
PubChem (143494026)
PubChem (162978898)
3E, F
(A, B)
waterwater18.058Chemie (HOH)
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains2
Total formula weight93701.0
Non-Polymers*Number of molecules2
Total formula weight933.1
All*Total formula weight94634.1
*Water molecules are not included.

251801

PDB entries from 2026-04-08

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