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4UVA

LSD1(KDM1A)-CoREST in complex with 1-Methyl-Tranylcypromine (1R,2S)

Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1ALYSINE-SPECIFIC HISTONE DEMETHYLASE 1Apolymer87294846.21UniProt (O60341)
Pfam (PF04433)
Pfam (PF01593)
In PDB
HOMO SAPIENS (HUMAN)BRAF35-HDAC COMPLEX PROTEIN BHC110, FLAVIN-CONTAINING AMINE OXIDASE DOMAIN-CONTAINING PROTEIN 2
2BREST COREPRESSOR 1polymer48253102.01UniProt (Q9UKL0)
Pfam (PF01448)
Pfam (PF00249)
Pfam (PF20878)
In PDB
HOMO SAPIENS (HUMAN)PROTEIN COREST
3A[(2R,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-3,4-dihydroxytetrahydrofuran-2-yl]methyl (2R,3S,4S)-2,3,4-trihydroxy-5-[(4aS)-4a-[(1S,3E)-3-imino-1-phenylbutyl]-7,8-dimethyl-2,4-dioxo-3,4,4a,5-tetrahydrobenzo[g]pteridin-10(2H)-yl]pentyl dihydrogen diphosphatenon-polymer932.81Chemie (D73)
4waterwater18.01Chemie (HOH)
Sequence modifications
A: -19 - 852 (UniProt: O60341)
PDBExternal DatabaseDetails
Pro 171Ala 191conflict
-Asp 390deletion
-Thr 391deletion
-Val 392deletion
-Lys 393deletion
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains2
Total formula weight147948.2
Non-Polymers*Number of molecules1
Total formula weight932.8
All*Total formula weight148881.0
*Water molecules are not included.

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PDB entries from 2024-09-18

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