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4S0T

STRUCTURE OF HUMAN PREGNANE X RECEPTOR LIGAND BINDING DOMAIN BOUND WITH ADNECTIN-1 AND COMPOUND-1

Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1A, BNuclear receptor subfamily 1 group I member 2polymer31536223.82UniProt (O75469)
Pfam (PF00104)
In PDB
Homo sapiens (human)Orphan nuclear receptor PAR1, Orphan nuclear receptor PXR, Pregnane X receptor, Steroid and xenobiotic receptor, SXR
2D, EAdnectin-1polymer12013232.62Homo sapiens (human)
3A, BN-{(2R)-1-[(4S)-4-(4-chlorophenyl)-4-hydroxy-3,3-dimethylpiperidin-1-yl]-3-methyl-1-oxobutan-2-yl}-2-cyclopropylacetamidenon-polymer421.02Chemie (40U)
Sequence modifications
A, B: 130 - 434 (UniProt: O75469)
PDBExternal DatabaseDetails
Met 120-expression tag
Lys 121-expression tag
Lys 122-expression tag
His 123-expression tag
His 124-expression tag
His 125-expression tag
His 126-expression tag
His 127-expression tag
His 128-expression tag
Gly 129-expression tag
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains4
Total formula weight98912.8
Non-Polymers*Number of molecules2
Total formula weight841.9
All*Total formula weight99754.8
*Water molecules are not included.

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PDB entries from 2024-06-12

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