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4S0T

STRUCTURE OF HUMAN PREGNANE X RECEPTOR LIGAND BINDING DOMAIN BOUND WITH ADNECTIN-1 AND COMPOUND-1

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006355biological_processregulation of DNA-templated transcription
B0003677molecular_functionDNA binding
B0004879molecular_functionnuclear receptor activity
B0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues10
DetailsBINDING SITE FOR RESIDUE 40U A 501
ChainResidue
AVAL211
AMET425
AMET243
AGLN285
APHE288
ATRP299
ATYR306
AMET323
AHIS407
APHE420

site_idAC2
Number of Residues12
DetailsBINDING SITE FOR RESIDUE 40U B 501
ChainResidue
BVAL211
BMET243
BALA244
BGLN285
BPHE288
BTRP299
BTYR306
BMET323
BHIS327
BHIS407
BPHE420
BMET425

Functional Information from PROSITE/UniProt
site_idPS00687
Number of Residues8
DetailsALDEHYDE_DEHYDR_GLU Aldehyde dehydrogenases glutamic acid active site. GETGGNSP
ChainResidueDetails
DGLY37-PRO44

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues6
DetailsBINDING: BINDING => ECO:0000269|PubMed:12578355, ECO:0007744|PDB:1M13
ChainResidueDetails
ASER247
AGLN285
AHIS407
BSER247
BGLN285
BHIS407

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PDB entries from 2024-07-31

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