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4Q9J

P-glycoprotein cocrystallised with QZ-Val

Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1AMultidrug resistance protein 1Apolymer1284141920.01UniProt (P21447)
Pfam (PF00664)
Pfam (PF00005)
In PDB
Mus musculus (mouse)ATP-binding cassette sub-family B member 1A, MDR1A, Multidrug resistance protein 3, P-glycoprotein 3
2C, D, BN-{[5-AMINO-1-(5-O-PHOSPHONO-BETA-D-ARABINOFURANOSYL)-1H-IMIDAZOL-4-YL]CARBONYL}-L-ASPARTIC ACIDpolymer6759.53BIRD (PRD_001235)
Sequence modifications
A: 1 - 1276 (UniProt: P21447)
PDBExternal DatabaseDetails
Gln 83Asn 83conflict
Gln 87Asn 87conflict
Gln 90Asn 90conflict
Leu 1277-expression tag
Glu 1278-expression tag
His 1279-expression tag
His 1280-expression tag
His 1281-expression tag
His 1282-expression tag
His 1283-expression tag
His 1284-expression tag
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains4
Total formula weight144198.4
All*Total formula weight144198.4
*Water molecules are not included.

217705

PDB entries from 2024-03-27

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