4Q9J
P-glycoprotein cocrystallised with QZ-Val
Entity
Entity ID | Chain ID | Description | Type | Chain length | Formula weight | Number of molecules | DB Name (Accession) | Biological source | Descriptive keywords |
1 | A | Multidrug resistance protein 1A | polymer | 1284 | 141920.0 | 1 | UniProt (P21447) Pfam (PF00664) Pfam (PF00005) In PDB | Mus musculus (mouse) | ATP-binding cassette sub-family B member 1A, MDR1A, Multidrug resistance protein 3, P-glycoprotein 3 |
2 | C, D, B | N-{[5-AMINO-1-(5-O-PHOSPHONO-BETA-D-ARABINOFURANOSYL)-1H-IMIDAZOL-4-YL]CARBONYL}-L-ASPARTIC ACID | polymer | 6 | 759.5 | 3 | BIRD (PRD_001235) |
Sequence modifications
A: 1 - 1276 (UniProt: P21447)
PDB | External Database | Details |
---|---|---|
Gln 83 | Asn 83 | conflict |
Gln 87 | Asn 87 | conflict |
Gln 90 | Asn 90 | conflict |
Leu 1277 | - | expression tag |
Glu 1278 | - | expression tag |
His 1279 | - | expression tag |
His 1280 | - | expression tag |
His 1281 | - | expression tag |
His 1282 | - | expression tag |
His 1283 | - | expression tag |
His 1284 | - | expression tag |
Sequence viewer
Contents of the asymmetric unit
Polymers | Number of chains | 4 |
Total formula weight | 144198.4 | |
All* | Total formula weight | 144198.4 |