4OLI
The pseudokinase/kinase protein from JAK-family member TYK2
Entity
Entity ID | Chain ID | Description | Type | Chain length | Formula weight | Number of molecules | DB Name (Accession) | Biological source | Descriptive keywords |
1 | A | Non-receptor tyrosine-protein kinase TYK2 | polymer | 645 | 73304.2 | 1 | UniProt (P29597) Pfam (PF07714) In PDB | Homo sapiens (human) | |
2 | A | 2-chloro-N-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}benzamide | non-polymer | 315.8 | 2 | Chemie (2TT) | |||
3 | water | water | 18.0 | 8 | Chemie (HOH) |
Sequence modifications
A: 566 - 1187 (UniProt: P29597)
PDB | External Database | Details |
---|---|---|
Met 543 | - | expression tag |
Ser 544 | - | expression tag |
Tyr 545 | - | expression tag |
Tyr 546 | - | expression tag |
His 547 | - | expression tag |
His 548 | - | expression tag |
His 549 | - | expression tag |
His 550 | - | expression tag |
His 551 | - | expression tag |
His 552 | - | expression tag |
Asp 553 | - | expression tag |
Tyr 554 | - | expression tag |
Asp 555 | - | expression tag |
Ile 556 | - | expression tag |
Pro 557 | - | expression tag |
Thr 558 | - | expression tag |
Thr 559 | - | expression tag |
Glu 560 | - | expression tag |
Asn 561 | - | expression tag |
Leu 562 | - | expression tag |
Tyr 563 | - | expression tag |
Phe 564 | - | expression tag |
Gln 565 | - | expression tag |
Ser 1016 | Ala 1016 | SEE REMARK 999 |
Asn 1023 | Asp 1023 | engineered mutation |
Sequence viewer
Contents of the asymmetric unit
Polymers | Number of chains | 1 |
Total formula weight | 73304.2 | |
Non-Polymers* | Number of molecules | 2 |
Total formula weight | 631.5 | |
All* | Total formula weight | 73935.7 |