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4LXD

Bcl_2-Navitoclax Analog (without Thiophenyl) Complex

Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1AApoptosis regulator Bcl-2polymer16619383.61UniProt (P10415)
Pfam (PF02180)
Pfam (PF00452)
In PDB
Homo sapiens (human)
2A4-(4-{[4-(4-chlorophenyl)-5,6-dihydro-2H-pyran-3-yl]methyl}piperazin-1-yl)-N-{[3-nitro-4-(tetrahydro-2H-pyran-4-ylamino)phenyl]sulfonyl}benzamidenon-polymer696.21Chemie (1XV)
3waterwater18.0231Chemie (HOH)
Sequence modifications
A: -1 - 32 (UniProt: P10415)
PDBExternal DatabaseDetails
Pro 2Ala 4engineered mutation
A: 89 - 204 (UniProt: P10415)
PDBExternal DatabaseDetails
Asp 73-linker
Val 74-linker
Glu 75-linker
Glu 76-linker
Asn 77-linker
Arg 78-linker
Thr 79-linker
Glu 80-linker
Ala 81-linker
Pro 82-linker
Glu 83-linker
Gly 84-linker
Thr 85-linker
Glu 86-linker
Ser 87-linker
Glu 88-linker
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains1
Total formula weight19383.6
Non-Polymers*Number of molecules1
Total formula weight696.2
All*Total formula weight20079.8
*Water molecules are not included.

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PDB entries from 2024-09-11

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