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4CFH

Structure of an active form of mammalian AMPK

Replaces:  2Y94
Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1A
(A)
5'-AMP-ACTIVATED PROTEIN KINASE CATALYTIC SUBUNIT ALPHA-1polymer49357248.51UniProt (P54645)
Pfam (PF00069)
Pfam (PF21147)
Pfam (PF16579)
RATTUS NORVEGICUS (NORWAY RAT)AMPK SUBUNIT ALPHA-1
2B
(B)
5'-AMP-ACTIVATED PROTEIN KINASE SUBUNIT BETA-2polymer8710040.81UniProt (O43741)
Pfam (PF04739)
HOMO SAPIENS (HUMAN)
3C
(C)
5'-AMP-ACTIVATED PROTEIN KINASE CATALYTIC SUBUNIT ALPHA-1polymer273064.61UniProt (P54645)RATTUS NORVEGICUS (NORWAY RAT)AMPK SUBUNIT ALPHA-1
4D
(E)
5'-AMP-ACTIVATED PROTEIN KINASE SUBUNIT GAMMA-1polymer33037434.11UniProt (P80385)
Pfam (PF00571)
RATTUS NORVEGICUS (NORWAY RAT)AMPK SUBUNIT ALPHA-1, AMPK GAMMA1, AMPK SUBUNIT GAMMA-1, AMPKG
5E
(A)
STAUROSPORINEnon-polymer466.51Chemie (STU)
PubChem (5279)
PubChem (44259)
PubChem (71203703)
PubChem (42610657)
PubChem (44299148)
PubChem (25322871)
PubChem (28684983)
PubChem (451705)
PubChem (44120114)
PubChem (44537813)
PubChem (49831000)
PubChem (46864193)
PubChem (68262703)
PubChem (68306294)
PubChem (5459111)
PubChem (73953205)
PubChem (6419748)
PubChem (86306248)
PubChem (358479)
PubChem (9804568)
PubChem (9937179)
PubChem (5280487)
PubChem (5311103)
PubChem (6711321)
PubChem (9956178)
PubChem (122130844)
PubChem (12046017)
PubChem (143163481)
PubChem (143224059)
PubChem (143494026)
PubChem (162978898)
6F, G
(E)
ADENOSINE MONOPHOSPHATEnon-polymer347.22Chemie (AMP)
PubChem (16397049)
PubChem (16760266)
PubChem (224)
PubChem (34768)
PubChem (83862)
PubChem (40467049)
PubChem (40469468)
PubChem (446048)
PubChem (44348067)
PubChem (45358029)
PubChem (40459109)
PubChem (515384)
PubChem (46874558)
PubChem (638042)
PubChem (46875232)
PubChem (57358045)
PubChem (57879893)
PubChem (57879902)
PubChem (5316444)
PubChem (5742864)
PubChem (177678969)
PubChem (6083)
PubChem (1549371)
PubChem (12163610)
PubChem (12358355)
PubChem (92144436)
PubChem (122197642)
PubChem (12358354)
PubChem (162290139)
PubChem (162946266)
PubChem (171699505)
Sequence modifications
A: 2 - 470 (UniProt: P54645)
PDBExternal DatabaseDetails
Met -18-expression tag
Ser -17-expression tag
His -16-expression tag
His -15-expression tag
His -14-expression tag
His -13-expression tag
His -12-expression tag
His -11-expression tag
Ser -10-expression tag
Ser -9-expression tag
Gly -8-expression tag
Leu -7-expression tag
Glu -6-expression tag
Val -5-expression tag
Leu -4-expression tag
Phe -3-expression tag
Gln -2-expression tag
Gly -1-expression tag
Pro 0-expression tag
Met 1-expression tag
Leu 471-SEE REMARK 999
Glu 472-SEE REMARK 999
Val 473-SEE REMARK 999
Leu 474-SEE REMARK 999
C: 524 - 548 (UniProt: P54645)
PDBExternal DatabaseDetails
Phe 522-SEE REMARK 999
Gln 523-SEE REMARK 999
B: 187 - 272 (UniProt: O43741)
PDBExternal DatabaseDetails
Met 186-expression tag
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains4
Total formula weight107788.0
Non-Polymers*Number of molecules3
Total formula weight1161.0
All*Total formula weight108949.0
*Water molecules are not included.

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PDB entries from 2026-04-01

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