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4CDR

Human O-GlcNAc transferase in complex with a bisubstrate inhibitor, Goblin1

Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1A, B, C, DUDP-N-ACETYLGLUCOSAMINE--PEPTIDE N-ACETYLGLUCOSAMINYLTRANSFERASE 110 KDA SUBUNITpolymer72380974.54UniProt (O15294)
Pfam (PF13424)
Pfam (PF13414)
Pfam (PF13844)
In PDB
HOMO SAPIENS (HUMAN)O-GLCNAC TRANSFERASE SUBUNIT P110, O-LINKED N-ACETYLGLUCOSAMINE TRANSFERASE 110 KDA SUBUNIT, OGT, O-GLCNAC TRANSFERASE
2E, F, G, HGOBLIN1polymer9755.94BIRD (PRD_002043)SYNTHETIC CONSTRUCT
3C, D, A, E, F...SULFATE IONnon-polymer96.131Chemie (SO4)
4E, F, G, HURIDINE-5'-DIPHOSPHATEnon-polymer404.24Chemie (UDP)
Sequence modifications
A, B, C, D: 313 - 1031 (UniProt: O15294)
PDBExternal DatabaseDetails
Gly 309-expression tag
Pro 310-expression tag
Gly 311-expression tag
Ser 312-expression tag
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains8
Total formula weight326921.5
Non-Polymers*Number of molecules35
Total formula weight4594.6
All*Total formula weight331516.1
*Water molecules are not included.

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PDB entries from 2024-08-07

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