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3PWH

Thermostabilised Adenosine A2A Receptor

Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1AAdenosine receptor A2apolymer32936479.11UniProt (P29274)
Pfam (PF00001)
In PDB
Homo sapiens (human)
2A4-{2-[(7-amino-2-furan-2-yl[1,2,4]triazolo[1,5-a][1,3,5]triazin-5-yl)amino]ethyl}phenolnon-polymer337.31Chemie (ZMA)
Sequence modifications
A: 1 - 317 (UniProt: P29274)
PDBExternal DatabaseDetails
Leu 54Ala 54engineered mutation
Ala 88Thr 88engineered mutation
Ala 107Arg 107engineered mutation
Ala 122Lys 122engineered mutation
Ala 202Leu 202engineered mutation
Ala 235Leu 235engineered mutation
Ala 239Val 239engineered mutation
Ala 277Ser 277engineered mutation
Ala 318-expression tag
Ala 319-expression tag
His 320-expression tag
His 321-expression tag
His 322-expression tag
His 323-expression tag
His 324-expression tag
His 325-expression tag
His 326-expression tag
His 327-expression tag
His 328-expression tag
His 329-expression tag
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains1
Total formula weight36479.1
Non-Polymers*Number of molecules1
Total formula weight337.3
All*Total formula weight36816.4
*Water molecules are not included.

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PDB entries from 2024-03-27

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