3JY9
Janus Kinase 2 Inhibitors
Entity
Entity ID | Chain ID | Description | Type | Chain length | Formula weight | Number of molecules | DB Name (Accession) | Biological source | Descriptive keywords |
1 | A | Tyrosine-protein kinase JAK2 | polymer | 311 | 36654.7 | 1 | UniProt (O60674) Pfam (PF07714) In PDB | Homo sapiens (human) | Janus kinase 2, JAK-2 |
2 | A | (3S)-3-(4-hydroxyphenyl)-1,5-dihydro-1,5,12-triazabenzo[4,5]cycloocta[1,2,3-cd]inden-4(3H)-one | non-polymer | 341.4 | 1 | Chemie (JZH) | |||
3 | A | SODIUM ION | non-polymer | 23.0 | 1 | Chemie (NA) | |||
4 | water | water | 18.0 | 176 | Chemie (HOH) |
Sequence modifications
A: 842 - 1130 (UniProt: O60674)
PDB | External Database | Details |
---|---|---|
Met 820 | - | expression tag |
Gly 821 | - | expression tag |
Ser 822 | - | expression tag |
Ser 823 | - | expression tag |
His 824 | - | expression tag |
His 825 | - | expression tag |
His 826 | - | expression tag |
His 827 | - | expression tag |
His 828 | - | expression tag |
His 829 | - | expression tag |
Ser 830 | - | expression tag |
Ser 831 | - | expression tag |
Gly 832 | - | expression tag |
Leu 833 | - | expression tag |
Val 834 | - | expression tag |
Pro 835 | - | expression tag |
Arg 836 | - | expression tag |
Gly 837 | - | expression tag |
Ser 838 | - | expression tag |
His 839 | - | expression tag |
Asn 840 | - | expression tag |
Met 841 | - | expression tag |
Sequence viewer
Contents of the asymmetric unit
Polymers | Number of chains | 1 |
Total formula weight | 36654.7 | |
Non-Polymers* | Number of molecules | 2 |
Total formula weight | 364.4 | |
All* | Total formula weight | 37019.0 |