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2X81

STRUCTURE OF AURORA A IN COMPLEX WITH MLN8054

Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1ASERINE/THREONINE-PROTEIN KINASE 6polymer27231440.21UniProt (O14965)
Pfam (PF00069)
In PDB
HOMO SAPIENS (HUMAN)AURORA A, AURORA KINASE A, SERINE/THREONINE-PROTEIN KINASE AURORA-A, SERINE/THREONINE-PROTEIN KINASE 15, AURORA/IPL1-RELATED KINASE 1, AURORA-RELATED KINASE 1, ARK-1, HARK1, BREAST TUMOR-AMPLIFIED KINASE
2A4-{[9-CHLORO-7-(2,6-DIFLUOROPHENYL)-5H-PYRIMIDO[5,4-D][2]BENZAZEPIN-2-YL]AMINO}BENZOIC ACIDnon-polymer476.91Chemie (ZZL)
Sequence modifications
A: 120 - 125 (PDB: 2X81)
A: 126 - 391 (UniProt: O14965)
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains1
Total formula weight31440.2
Non-Polymers*Number of molecules1
Total formula weight476.9
All*Total formula weight31917.0
*Water molecules are not included.

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PDB entries from 2024-09-18

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