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2EWA

Dual binding mode of pyridinylimidazole to MAP kinase p38

Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1AMitogen-activated protein kinase 14polymer37943383.41UniProt (P47811)
Pfam (PF00069)
In PDB
Mus musculus (house mouse)Mitogen-activated protein kinase p38 alpha, MAP kinase p38 alpha, CRK1
2A4-[5-(4-FLUORO-PHENYL)-2-(4-METHANESULFINYL-PHENYL)-3H-IMIDAZOL-4-YL]-PYRIDINEnon-polymer377.41Chemie (SB2)
3waterwater18.073Chemie (HOH)
Sequence modifications
A: 1 - 360 (UniProt: P47811)
PDBExternal DatabaseDetails
Gly -18-cloning artifact
Ser -17-cloning artifact
Ser -16-cloning artifact
His -15-expression tag
His -14-expression tag
His -13-expression tag
His -12-expression tag
His -11-expression tag
His -10-expression tag
Ser -9-cloning artifact
Ser -8-cloning artifact
Gly -7-cloning artifact
Leu -6-cloning artifact
Val -5-cloning artifact
Pro -4-cloning artifact
Arg -3-cloning artifact
Gly -2-cloning artifact
Ser -1-cloning artifact
His 0-cloning artifact
Leu 48His 47conflict
Thr 263Ala 262conflict
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains1
Total formula weight43383.4
Non-Polymers*Number of molecules1
Total formula weight377.4
All*Total formula weight43760.8
*Water molecules are not included.

222036

PDB entries from 2024-07-03

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