2BZ6
Orally available Factor7a inhibitor
Entity
Entity ID | Chain ID | Description | Type | Chain length | Formula weight | Number of molecules | DB Name (Accession) | Biological source | Descriptive keywords |
1 | A (H) | BLOOD COAGULATION FACTOR VIIA | polymer | 254 | 28103.3 | 1 | UniProt (P08709) Pfam (PF00089) | HOMO SAPIENS (HUMAN) | SERUM PROTHROMBIN CONVERSION ACCELERATOR, SPCA, PROCONVERTIN, EPTACOG ALFA, NOVOSEVEN |
2 | B (L) | BLOOD COAGULATION FACTOR VIIA | polymer | 53 | 5744.5 | 1 | UniProt (P08709) Pfam (PF14670) | HOMO SAPIENS (HUMAN) | SERUM PROTHROMBIN CONVERSION ACCELERATOR, SPCA, PROCONVERTIN, EPTACOG ALFA, NOVOSEVEN |
3 | C (H) | (R)-(4-CARBAMIMIDOYL-PHENYLAMINO)-[5-ETHOXY-2-FLUORO-3-[(R)-TETRAHYDRO-FURAN-3-YLOXY]-PHENYL]-ACETIC ACID | non-polymer | 417.4 | 1 | Chemie (346) | |||
4 | D (H) | SULFATE ION | non-polymer | 96.1 | 1 | Chemie (SO4) | |||
5 | E (H) | CALCIUM ION | non-polymer | 40.1 | 1 | Chemie (CA) | |||
6 | F, G (H, L) | water | water | 18.0 | 500 | Chemie (HOH) |
Sequence viewer
Contents of the asymmetric unit
Polymers | Number of chains | 2 |
Total formula weight | 33847.7 | |
Non-Polymers* | Number of molecules | 3 |
Total formula weight | 553.6 | |
All* | Total formula weight | 34401.3 |