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1S1T

Crystal structure of L100I mutant HIV-1 reverse transcriptase in complex with UC-781

Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1AReverse transcriptasepolymer56064594.91UniProt (P04585)
Pfam (PF00078)
Pfam (PF06817)
Pfam (PF06815)
Pfam (PF00075)
In PDB
Human immunodeficiency virus 1HIV-1 RT
2BReverse transcriptasepolymer44051399.01UniProt (P04585)
Pfam (PF00078)
Pfam (PF06817)
Pfam (PF06815)
In PDB
Human immunodeficiency virus 1HIV-1 RT
3A, BPHOSPHATE IONnon-polymer95.02Chemie (PO4)
4A2-METHYL-FURAN-3-CARBOTHIOIC ACID [4-CHLORO-3-(3-METHYL-BUT-2-ENYLOXY)-PHENYL]-AMIDEnon-polymer335.81Chemie (UC1)
5waterwater18.0184Chemie (HOH)
Sequence modifications
A: 1 - 560 (UniProt: P04585)
PDBExternal DatabaseDetails
Ile 100Leu 255engineered mutation
Csd 280Cys 435modified residue
B: 1 - 440 (UniProt: P04585)
PDBExternal DatabaseDetails
Ile 100Leu 255engineered mutation
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains2
Total formula weight115994.0
Non-Polymers*Number of molecules3
Total formula weight525.8
All*Total formula weight116519.8
*Water molecules are not included.

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PDB entries from 2024-09-18

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