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1FVV

THE STRUCTURE OF CDK2/CYCLIN A IN COMPLEX WITH AN OXINDOLE INHIBITOR

Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1A, CCYCLIN-DEPENDENT KINASE 2polymer29833976.52UniProt (P24941)
Pfam (PF00069)
In PDB
Homo sapiens (human)CDK2, P33 PROTEIN KINASE
2B, DCYCLIN Apolymer26029867.52UniProt (P20248)
Pfam (PF00134)
Pfam (PF02984)
In PDB
Homo sapiens (human)CYCLIN A2
3A, C4-[(7-OXO-7H-THIAZOLO[5,4-E]INDOL-8-YLMETHYL)-AMINO]-N-PYRIDIN-2-YL-BENZENESULFONAMIDEnon-polymer449.52Chemie (107)
4waterwater18.0129Chemie (HOH)
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains4
Total formula weight127688.0
Non-Polymers*Number of molecules2
Total formula weight899.0
All*Total formula weight128587.0
*Water molecules are not included.

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PDB entries from 2024-04-24

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