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5IBQ
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Crystal structure of an ABC solute binding protein from Rhizobium etli CFN 42 (RHE_PF00037,TARGET EFI-511357) in complex with alpha-D-apiose
分子名称: 3-C-(hydroxylmethyl)-alpha-D-erythrofuranose, CALCIUM ION, Probable ribose ABC transporter, ...
著者Vetting, M.W, Carter, M.S, Al Obaidi, N.F, Morisco, L.L, Benach, J, Koss, J, Wasserman, S.R, Gerlt, J.A, Almo, S.C, Enzyme Function Initiative (EFI)
登録日2016-02-22
公開日2016-04-20
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.2 Å)
主引用文献Crystal structure of an ABC solute binding protein from Rhizobium etli CFN 42 (RHE_PF00037,TARGET EFI-511357) in complex with alpha-D-apiose
To be published
2BKS
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BU of 2bks by Molmil
crystal structure of Renin-PF00074777 complex
分子名称: (6R)-6-({[1-(3-HYDROXYPROPYL)-1,7-DIHYDROQUINOLIN-7-YL]OXY}METHYL)-1-(4-{3-[(2-METHOXYBENZYL)OXY]PROPOXY}PHENYL)PIPERAZIN-2-ONE, Renin
著者Powell, N.A, Clay, E.H, Holsworth, D.D, Edmunds, J.J, Bryant, J.W, Ryan, J.M, Jalaie, M, Zhang, E.
登録日2005-02-18
公開日2006-04-05
最終更新日2021-07-21
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Equipotent Activity in Both Enantiomers of a Series of Ketopiperazine-Based Renin Inhibitors
Bioorg.Med.Chem.Lett., 15, 2005
4UJ1
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Protein Kinase A in complex with an Inhibitor
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, 7-[(3S,4R)-4-(3-chlorophenyl)carbonylpyrrolidin-3-yl]-3H-quinazolin-4-one, CAMP-DEPENDENT PROTEIN KINASE CATALYTIC SUBUNIT ALPHA, ...
著者Alam, K.A, Engh, R.A.
登録日2015-04-07
公開日2016-04-13
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.768 Å)
主引用文献Addressing the Glycine-Rich Loop of Protein Kinases by a Multi-Facetted Interaction Network: Inhibition of Pka and a Pkb Mimic.
Chemistry, 22, 2016
4USE
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BU of 4use by Molmil
Human STK10 (LOK) with SB-633825
分子名称: 4-{5-(6-methoxynaphthalen-2-yl)-1-methyl-2-[2-methyl-4-(methylsulfonyl)phenyl]-1H-imidazol-4-yl}pyridine, SERINE/THREONINE-PROTEIN KINASE 10
著者Elkins, J.M, Salah, E, Szklarz, M, von Delft, F, Canning, P, Raynor, J, Bountra, C, Edwards, A.M, Knapp, S.
登録日2014-07-07
公開日2015-07-22
最終更新日2018-01-24
実験手法X-RAY DIFFRACTION (2.65 Å)
主引用文献Comprehensive Characterization of the Published Kinase Inhibitor Set.
Nat.Biotechnol., 34, 2016
4V0M
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BU of 4v0m by Molmil
Crystal structure of BBS1N in complex with ARL6DN
分子名称: ARF-LIKE SMALL GTPASE, BARDET-BIEDL SYNDROME 1 PROTEIN, GUANOSINE-5'-TRIPHOSPHATE, ...
著者Mourao, A, Lorentzen, E.
登録日2014-09-17
公開日2014-11-19
最終更新日2019-04-03
実験手法X-RAY DIFFRACTION (3.45 Å)
主引用文献Structural Basis for Membrane Targeting of the Bbsome by Arl6
Nat.Struct.Mol.Biol., 21, 2014
4LIJ
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BU of 4lij by Molmil
Crystal structure of a far upstream element (FUSE) binding protein 1 (FUBP1) from Homo sapiens at 1.95 A resolution
分子名称: Far upstream element-binding protein 1, PHOSPHATE ION
著者Joint Center for Structural Genomics (JCSG), Partnership for T-Cell Biology, Partnership for T-Cell Biology (TCELL)
登録日2013-07-02
公開日2013-11-27
最終更新日2023-02-01
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Crystal structure of a far upstream element (FUSE) binding protein 1 (FUBP1) from Homo sapiens at 1.95 A resolution
To be published
9CTX
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BU of 9ctx by Molmil
X-ray crystal structure of multi-drug resistant HIV-1 protease (P51) in complex with Darunavir
分子名称: (3R,3AS,6AR)-HEXAHYDROFURO[2,3-B]FURAN-3-YL(1S,2R)-3-[[(4-AMINOPHENYL)SULFONYL](ISOBUTYL)AMINO]-1-BENZYL-2-HYDROXYPROPYLCARBAMATE, GLYCEROL, Protease
著者Hayashi, H, Yedidi, R, Bulut, H, Das, D, Mitsuya, H.
登録日2024-07-25
公開日2024-08-07
実験手法X-RAY DIFFRACTION (1.55 Å)
主引用文献Secondary amino-acid substitutions contribute to the emergence of HIV protease inhibitor resistance as directly as primary amino-acid substitutions.
To Be Published
9GEA
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Structure of UP1 S4DS6D phosphomimetic mutant
分子名称: Heterogeneous nuclear ribonucleoprotein A1, N-terminally processed
著者Dunnett, L, Prischi, F.
登録日2024-08-07
公開日2024-08-21
実験手法X-RAY DIFFRACTION (1.89 Å)
主引用文献Structure of UP1 S4DS6D phosphomimetic mutant
To Be Published
9G11
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BU of 9g11 by Molmil
sugar/H+ symporter STP6 in inward occluded conformation with glucose bound
分子名称: CHOLESTEROL HEMISUCCINATE, Sugar transport protein 6, beta-D-glucopyranose
著者Andersen, C.G, Bavnhoj, L, Pedersen, B.P.
登録日2024-07-09
公開日2024-08-14
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Comparative biochemical analysis of the plant sugar transporters STP6 and STP10
To Be Published
7O0K
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BU of 7o0k by Molmil
Crystal structure of recombinant chichen liver Bile Acid Binding Protein (cL-BABP) in complex with cholic acid
分子名称: CHOLIC ACID, Fatty acid-binding protein, liver
著者Tassone, G, Pozzi, C.
登録日2021-03-26
公開日2021-05-12
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.83 Å)
主引用文献Validation of Recombinant Chicken Liver Bile Acid Binding Protein as a Tool for Cholic Acid Hosting.
Biomolecules, 11, 2021
7O0J
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High resolution structure of recombinant chichen liver Bile Acid Binding Protein (cL-BABP)
分子名称: Fatty acid-binding protein, liver
著者Tassone, G, Pozzi, C.
登録日2021-03-26
公開日2021-05-12
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献Validation of Recombinant Chicken Liver Bile Acid Binding Protein as a Tool for Cholic Acid Hosting.
Biomolecules, 11, 2021
7NUM
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BU of 7num by Molmil
Rhinovirus-14 ICAM-1 empty particle at pH 6.2
分子名称: Genome polyprotein, P1
著者Hrebik, D, Plevka, P.
登録日2021-03-12
公開日2021-05-19
最終更新日2024-07-10
実験手法ELECTRON MICROSCOPY (3.9 Å)
主引用文献ICAM-1 induced rearrangements of capsid and genome prime rhinovirus 14 for activation and uncoating.
Proc.Natl.Acad.Sci.USA, 118, 2021
7NUO
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Rhinovirus 14 empty particle at pH 6.2
分子名称: Genome polyprotein, P1
著者Hrebik, D, Plevka, P.
登録日2021-03-12
公開日2021-05-19
最終更新日2024-07-10
実験手法ELECTRON MICROSCOPY (3.9 Å)
主引用文献ICAM-1 induced rearrangements of capsid and genome prime rhinovirus 14 for activation and uncoating.
Proc.Natl.Acad.Sci.USA, 118, 2021
7OAJ
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BU of 7oaj by Molmil
Crystal structure of pseudokinase CASK in complex with compound 7
分子名称: 1,2-ETHANEDIOL, 4-(cyclopentylamino)-2-[(3,4-dichlorophenyl)methylamino]-N-[3-(2-oxidanylidenepyrrolidin-1-yl)propyl]pyrimidine-5-carboxamide, Peripheral plasma membrane protein CASK
著者Chaikuad, A, Russ, N, Knapp, S, Structural Genomics Consortium (SGC)
登録日2021-04-19
公開日2021-05-19
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.93 Å)
主引用文献Design and Development of a Chemical Probe for Pseudokinase Ca 2+ /calmodulin-Dependent Ser/Thr Kinase.
J.Med.Chem., 64, 2021
7OAI
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BU of 7oai by Molmil
Crystal structure of pseudokinase CASK in complex with PFE-PKIS12
分子名称: 1,2-ETHANEDIOL, 4-(Cyclopentylamino)-2-[(2,5-dichlorophenyl)methylamino]-N-[3-(2-oxo-1,3-oxazolidin-3-yl)propyl]pyrimidine-5-carboxamide, Peripheral plasma membrane protein CASK
著者Chaikuad, A, Knapp, S, Structural Genomics Consortium (SGC)
登録日2021-04-19
公開日2021-05-19
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Design and Development of a Chemical Probe for Pseudokinase Ca 2+ /calmodulin-Dependent Ser/Thr Kinase.
J.Med.Chem., 64, 2021
7NUL
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BU of 7nul by Molmil
Rhinovirus-14 ICAM-1 activated particle at pH 6.2
分子名称: Genome polyprotein, P1
著者Hrebik, D, Plevka, P.
登録日2021-03-12
公開日2021-05-19
最終更新日2024-07-10
実験手法ELECTRON MICROSCOPY (4 Å)
主引用文献ICAM-1 induced rearrangements of capsid and genome prime rhinovirus 14 for activation and uncoating.
Proc.Natl.Acad.Sci.USA, 118, 2021
7OAK
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BU of 7oak by Molmil
Crystal structure of pseudokinase CASK in complex with compound 26
分子名称: 1,2-ETHANEDIOL, 2-[[2,5-bis(bromanyl)-4-methyl-phenyl]methylamino]-4-(cyclopentylamino)-N-[3-(2-oxidanylidene-1,3-oxazolidin-3-yl)propyl]pyrimidine-5-carboxamide, Peripheral plasma membrane protein CASK
著者Chaikuad, A, Russ, N, Knapp, S, Structural Genomics Consortium (SGC)
登録日2021-04-19
公開日2021-05-19
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.23 Å)
主引用文献Design and Development of a Chemical Probe for Pseudokinase Ca 2+ /calmodulin-Dependent Ser/Thr Kinase.
J.Med.Chem., 64, 2021
7OAL
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BU of 7oal by Molmil
Crystal structure of pseudokinase CASK in complex with compound 25
分子名称: 1,2-ETHANEDIOL, 2-[[2,5-bis(bromanyl)-4-methyl-phenyl]methylamino]-4-(cyclohexylamino)-N-[3-(2-oxidanylidene-1,3-oxazolidin-3-yl)propyl]pyrimidine-5-carboxamide, Peripheral plasma membrane protein CASK
著者Chaikuad, A, Russ, N, Knapp, S, Structural Genomics Consortium (SGC)
登録日2021-04-19
公開日2021-05-19
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.17 Å)
主引用文献Design and Development of a Chemical Probe for Pseudokinase Ca 2+ /calmodulin-Dependent Ser/Thr Kinase.
J.Med.Chem., 64, 2021
7NXE
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BU of 7nxe by Molmil
Structure of the Phospholipase C gamma 1 tSH2 domain in complex with a phosphorylated KSHV pK15 peptide
分子名称: Isoform 2 of 1-phosphatidylinositol 4,5-bisphosphate phosphodiesterase gamma-1, Protein K15
著者Ssebyatika, G, Krey, T.
登録日2021-03-18
公開日2021-06-09
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Recruitment of phospholipase C gamma 1 to the non-structural membrane protein pK15 of Kaposi Sarcoma-associated herpesvirus promotes its Src-dependent phosphorylation.
Plos Pathog., 17, 2021
7NVQ
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BU of 7nvq by Molmil
Aerosol-soaked human cdk2 crystals with Staurosporine
分子名称: 1,2-ETHANEDIOL, Cyclin-dependent kinase 2, STAUROSPORINE
著者Ross, B, Huber, R.
登録日2021-03-15
公開日2021-06-16
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献Aerosol-based ligand soaking of reservoir-free protein crystals.
J.Appl.Crystallogr., 54, 2021
7NY8
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BU of 7ny8 by Molmil
Affimer K69 - KRAS protein complex
分子名称: Affimer K69, GTPase KRas, GUANOSINE-5'-DIPHOSPHATE, ...
著者Turner, A.L, Trinh, C.H, Haza, K.Z, Rao, A, Martin, H.L, Tiede, C, Edwards, T.A, McPherson, M.J, Tomlinson, D.C.
登録日2021-03-21
公開日2021-07-07
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献RAS-inhibiting biologics identify and probe druggable pockets including an SII-alpha 3 allosteric site.
Nat Commun, 12, 2021
8BKH
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BU of 8bkh by Molmil
Carboxymyoglobin dark state for comparison with power titration and 23 / 101 mJ/cm2 time series
分子名称: CARBON MONOXIDE, Myoglobin, PROTOPORPHYRIN IX CONTAINING FE, ...
著者Barends, T, Schlichting, I.
登録日2022-11-09
公開日2024-01-31
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (1.35 Å)
主引用文献Influence of pump laser fluence on ultrafast myoglobin structural dynamics.
Nature, 626, 2024
8BKN
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Carboxymyoglobin dark state for comparison with 5 mJ/cm2 time series
分子名称: CARBON MONOXIDE, Myoglobin, PROTOPORPHYRIN IX CONTAINING FE, ...
著者Barends, T, Schlichting, I.
登録日2022-11-09
公開日2024-01-31
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (1.29 Å)
主引用文献Influence of pump laser fluence on ultrafast myoglobin structural dynamics.
Nature, 626, 2024
8BWN
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Crystal structure of human Twisted gastrulation protein homolog 1 (TWSG1) in complex with human Growth Differentiation Factor 5 (GDF5) and calcium, long-wavelength X-ray dataset (4010 eV)
分子名称: CALCIUM ION, Growth/differentiation factor 5, Twisted gastrulation protein homolog 1
著者Malinauskas, T, Rudolf, A.F, Moore, G, Eggington, H, Belnoue-Davis, H, El Omari, K, Woolley, R.E, Griffiths, S.C, Duman, R, Wagner, A, Leedham, S.J, Baldock, C, Ashe, H, Siebold, C.
登録日2022-12-07
公開日2024-06-19
実験手法X-RAY DIFFRACTION (2.57 Å)
主引用文献Molecular mechanism of BMP signal control by Twisted gastrulation.
Nat Commun, 15, 2024
8BWL
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Crystal structure of human Twisted gastrulation protein homolog 1 (TWSG1) in complex with human Growth Differentiation factor 5 (GDF5) and calcium
分子名称: CALCIUM ION, Growth/differentiation factor 5, Twisted gastrulation protein homolog 1
著者Malinauskas, T, Rudolf, A.F, Moore, G, Eggington, H, Belnoue-Davis, H, El Omari, K, Woolley, R.E, Griffiths, S.C, Duman, R, Wagner, A, Leedham, S.J, Baldock, C, Ashe, H, Siebold, C.
登録日2022-12-06
公開日2024-06-19
実験手法X-RAY DIFFRACTION (1.96 Å)
主引用文献Molecular mechanism of BMP signal control by Twisted gastrulation.
Nat Commun, 15, 2024

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