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9KGR

Discovery of an orally bioavailable reversible covalent SARS-CoV-2 Mpro inhibitor with pan-coronavirus activity

This is a non-PDB format compatible entry.
Resources
File formatFile name (file size)
PDBx/mmCIF9kgr.cif.gz Display(172.91 KB)
9kgr.cif
PDBx/mmJSONall9kgr.json.gz Display (Tree)(119.34 KB)
9kgr.json
no-atom9kgr-noatom.json.gz Display (Header)(18.51 KB)
9kgr-noatom.json
add only9kgr-plus.json.gz Display(788.00 B)
9kgr-plus.json
PDBMLall9kgr.xml.gz Display(219.66 KB)
9kgr.xml
no-atom9kgr-noatom.xml.gz Display(36.98 KB)
9kgr-noatom.xml
ext-atom9kgr-extatom.xml.gz Display(143.69 KB)
9kgr-extatom.xml
pdb_nextgenallpdb_00009kgr_xyz-enrich.cif.gz Display(188.19 KB)
pdb_00009kgr_xyz-enrich.cif
no-atompdb_00009kgr_xyz-no-atom-enrich.xml.gz Display(49.27 KB)
pdb_00009kgr_xyz-no-atom-enrich.xml
ng-only9kgr-plus.json.gz Display(3.25 KB)
9kgr-plus.json
RDF9kgr.rdf.gz Visualize(104.79 KB)
9kgr.rdf
Structure factorsr9kgrsf.ent.gz Display(3.26 MB)
r9kgrsf.ent
Biological unit (mmCIF format)9kgr-assembly1.cif.gz Display(141.73 KB)
9kgr-assembly1.cif (A,B,C,D)

*author and software defined assembly, 4 molecule(s) (tetrameric)

Validation reportsPDF9kgr_validation.pdf.gz Display(1.01 MB)
9kgr_validation.pdf
PDF-full9kgr_full_validation.pdf.gz Display(1.01 MB)
9kgr_full_validation.pdf
mmCIF9kgr_validation.cif.gz Display(45.03 KB)
9kgr_validation.cif
XML9kgr_validation.xml.gz Display(32.29 KB)
9kgr_validation.xml
PNG9kgr_multipercentile_validation.png.gz Display(163.16 KB)
9kgr_multipercentile_validation.png
SVG9kgr_multipercentile_validation.svg.gz Display(921.00 B)
9kgr_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)9kgr_validation_2fo-fc_map_coef.cif.gz Display(1.34 MB)
9kgr_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)9kgr_validation_fo-fc_map_coef.cif.gz Display(1.34 MB)
9kgr_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)9kgr_validation_2fo-fc_map_coef.mtz Visualize(2.11 MB)
fo-fc (MTZ)9kgr_validation_fo-fc_map_coef.mtz Visualize(2.11 MB)

243083

PDB entries from 2025-10-15

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