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8STG

Discovery and clinical validation of RLY-4008, the first highly selective FGFR2 inhibitor with activity across FGFR2 alterations and resistance mutations

Resources
File formatFile name (file size)
PDBx/mmCIF8stg.cif.gz Display(267.66 KB)
8stg.cif
PDBx/mmJSONall8stg.json.gz Display (Tree)(187.68 KB)
8stg.json
no-atom8stg-noatom.json.gz Display (Header)(17.78 KB)
8stg-noatom.json
add only8stg-plus.json.gz Display(1.11 KB)
8stg-plus.json
PDBMLall8stg.xml.gz Display(335.03 KB)
8stg.xml
no-atom8stg-noatom.xml.gz Display(32.35 KB)
8stg-noatom.xml
ext-atom8stg-extatom.xml.gz Display(236.50 KB)
8stg-extatom.xml
PDBpdb8stg.ent.gz Display(176.19 KB)
pdb8stg.ent
RDF8stg.rdf.gz Visualize(96.09 KB)
8stg.rdf
Structure factorsr8stgsf.ent.gz Display(220.75 KB)
r8stgsf.ent
Biological unit (mmCIF format)8stg-assembly1.cif.gz Display(114.38 KB)
8stg-assembly1.cif (A)

*author defined assembly, 1 molecule(s) (monomeric)

8stg-assembly2.cif.gz Display(114.79 KB)
8stg-assembly2.cif (B)

*author defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)8stg.pdb1.gz Display(86.89 KB)
8stg.pdb1 (A)

*author defined assembly, 1 molecule(s) (monomeric)

8stg.pdb2.gz Display(86.60 KB)
8stg.pdb2 (B)

*author defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF8stg_validation.pdf.gz Display(1009.30 KB)
8stg_validation.pdf
PDF-full8stg_full_validation.pdf.gz Display(1.00 MB)
8stg_full_validation.pdf
mmCIF8stg_validation.cif.gz Display(30.81 KB)
8stg_validation.cif
XML8stg_validation.xml.gz Display(23.80 KB)
8stg_validation.xml
PNG8stg_multipercentile_validation.png.gz Display(170.15 KB)
8stg_multipercentile_validation.png
SVG8stg_multipercentile_validation.svg.gz Display(955.00 B)
8stg_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)8stg_validation_2fo-fc_map_coef.cif.gz Display(78.02 KB)
8stg_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)8stg_validation_fo-fc_map_coef.cif.gz Display(77.16 KB)
8stg_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)8stg_validation_2fo-fc_map_coef.mtz Visualize(185.98 KB)
fo-fc (MTZ)8stg_validation_fo-fc_map_coef.mtz Visualize(185.98 KB)

223166

PDB entries from 2024-07-31

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