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8ENJ

Design, synthesis, biological evaluation, and X-ray crystallography of diarylpyrazole derivatives possessing terminal arylsulfonamide moieties as anti-proliferative agents targeting c-Jun N-terminal kinase (JNK)

Resources
File formatFile name (file size)
PDBx/mmCIF8enj.cif.gz Display(183.02 KB)
8enj.cif
PDBx/mmJSONall8enj.json.gz Display (Tree)(136.46 KB)
8enj.json
no-atom8enj-noatom.json.gz Display (Header)(18.77 KB)
8enj-noatom.json
add only8enj-plus.json.gz Display(1.21 KB)
8enj-plus.json
PDBMLall8enj.xml.gz Display(234.20 KB)
8enj.xml
no-atom8enj-noatom.xml.gz Display(30.44 KB)
8enj-noatom.xml
ext-atom8enj-extatom.xml.gz Display(77.25 KB)
8enj-extatom.xml
PDBpdb8enj.ent.gz Display(120.27 KB)
pdb8enj.ent
RDF8enj.rdf.gz Visualize(91.01 KB)
8enj.rdf
Structure factorsr8enjsf.ent.gz Display(272.63 KB)
r8enjsf.ent
Biological unit (mmCIF format)8enj-assembly1.cif.gz Display(158.74 KB)
8enj-assembly1.cif (A)

*author defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)8enj.pdb1.gz Display(113.88 KB)
8enj.pdb1 (A)

*author defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF8enj_validation.pdf.gz Display(805.34 KB)
8enj_validation.pdf
PDF-full8enj_full_validation.pdf.gz Display(821.86 KB)
8enj_full_validation.pdf
mmCIF8enj_validation.cif.gz Display(21.74 KB)
8enj_validation.cif
XML8enj_validation.xml.gz Display(16.91 KB)
8enj_validation.xml
PNG8enj_multipercentile_validation.png.gz Display(167.04 KB)
8enj_multipercentile_validation.png
SVG8enj_multipercentile_validation.svg.gz Display(972.00 B)
8enj_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)8enj_validation_2fo-fc_map_coef.cif.gz Display(101.17 KB)
8enj_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)8enj_validation_fo-fc_map_coef.cif.gz Display(99.41 KB)
8enj_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)8enj_validation_2fo-fc_map_coef.mtz Visualize(242.87 KB)
fo-fc (MTZ)8enj_validation_fo-fc_map_coef.mtz Visualize(242.87 KB)

222415

PDB entries from 2024-07-10

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