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8DEA

Scaffold Hopping via Ring Opening Enables Identification of Acyclic Compounds as New Complement Factor D Inhibitors

Resources
File formatFile name (file size)
PDBx/mmCIF8dea.cif.gz Display(182.05 KB)
8dea.cif
PDBx/mmJSONall8dea.json.gz Display (Tree)(117.10 KB)
8dea.json
no-atom8dea-noatom.json.gz Display (Header)(17.28 KB)
8dea-noatom.json
add only8dea-plus.json.gz Display(1.05 KB)
8dea-plus.json
PDBMLall8dea.xml.gz Display(249.23 KB)
8dea.xml
no-atom8dea-noatom.xml.gz Display(38.80 KB)
8dea-noatom.xml
ext-atom8dea-extatom.xml.gz Display(153.90 KB)
8dea-extatom.xml
PDBpdb8dea.ent.gz Display(138.99 KB)
pdb8dea.ent
RDF8dea.rdf.gz Visualize(109.63 KB)
8dea.rdf
Structure factorsr8deasf.ent.gz Display(1.08 MB)
r8deasf.ent
Biological unit (mmCIF format)8dea-assembly1.cif.gz Display(46.64 KB)
8dea-assembly1.cif (A)

*author defined assembly, 1 molecule(s) (monomeric)

8dea-assembly2.cif.gz Display(46.55 KB)
8dea-assembly2.cif (B)

*author defined assembly, 1 molecule(s) (monomeric)

8dea-assembly3.cif.gz Display(47.19 KB)
8dea-assembly3.cif (C)

*author defined assembly, 1 molecule(s) (monomeric)

8dea-assembly4.cif.gz Display(46.70 KB)
8dea-assembly4.cif (D)

*author defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)8dea.pdb1.gz Display(35.46 KB)
8dea.pdb1 (A)

*author defined assembly, 1 molecule(s) (monomeric)

8dea.pdb2.gz Display(35.84 KB)
8dea.pdb2 (B)

*author defined assembly, 1 molecule(s) (monomeric)

8dea.pdb3.gz Display(35.96 KB)
8dea.pdb3 (C)

*author defined assembly, 1 molecule(s) (monomeric)

8dea.pdb4.gz Display(35.75 KB)
8dea.pdb4 (D)

*author defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF8dea_validation.pdf.gz Display(1.59 MB)
8dea_validation.pdf
PDF-full8dea_full_validation.pdf.gz Display(1.60 MB)
8dea_full_validation.pdf
mmCIF8dea_validation.cif.gz Display(44.81 KB)
8dea_validation.cif
XML8dea_validation.xml.gz Display(33.81 KB)
8dea_validation.xml
PNG8dea_multipercentile_validation.png.gz Display(165.93 KB)
8dea_multipercentile_validation.png
SVG8dea_multipercentile_validation.svg.gz Display(974.00 B)
8dea_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)8dea_validation_2fo-fc_map_coef.cif.gz Display(397.10 KB)
8dea_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)8dea_validation_fo-fc_map_coef.cif.gz Display(362.46 KB)
8dea_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)8dea_validation_2fo-fc_map_coef.mtz Visualize(954.62 KB)
fo-fc (MTZ)8dea_validation_fo-fc_map_coef.mtz Visualize(954.62 KB)

222415

PDB entries from 2024-07-10

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