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7U4R

Structure of MAP kinase phosphatase 5 in complex with 3,3-dimethyl-1-((9-propyl-5,6-dihydrothieno[2,3-h]quinazolin-2-yl)thio)butan-2-one, an allosteric inhibitor

Resources
File formatFile name (file size)
PDBx/mmCIF7u4r.cif.gz Display(445.96 KB)
7u4r.cif
PDBx/mmJSONall7u4r.json.gz Display (Tree)(311.63 KB)
7u4r.json
no-atom7u4r-noatom.json.gz Display (Header)(23.08 KB)
7u4r-noatom.json
add only7u4r-plus.json.gz Display(1.07 KB)
7u4r-plus.json
PDBMLall7u4r.xml.gz Display(582.39 KB)
7u4r.xml
no-atom7u4r-noatom.xml.gz Display(45.23 KB)
7u4r-noatom.xml
ext-atom7u4r-extatom.xml.gz Display(203.11 KB)
7u4r-extatom.xml
pdb_nextgenallpdb_00007u4r_xyz-enrich.cif.gz Display(464.80 KB)
pdb_00007u4r_xyz-enrich.cif
no-atompdb_00007u4r_xyz-no-atom-enrich.xml.gz Display(66.31 KB)
pdb_00007u4r_xyz-no-atom-enrich.xml
ng-only7u4r-plus.json.gz Display(2.57 KB)
7u4r-plus.json
PDBpdb7u4r.ent.gz Display(311.90 KB)
pdb7u4r.ent
RDF7u4r.rdf.gz Visualize(112.99 KB)
7u4r.rdf
Structure factorsr7u4rsf.ent.gz Display(762.34 KB)
r7u4rsf.ent
Biological unit (mmCIF format)7u4r-assembly1.cif.gz Display(73.07 KB)
7u4r-assembly1.cif (A)

*author defined assembly, 1 molecule(s) (monomeric)

7u4r-assembly2.cif.gz Display(72.87 KB)
7u4r-assembly2.cif (B)

*author defined assembly, 1 molecule(s) (monomeric)

7u4r-assembly3.cif.gz Display(72.73 KB)
7u4r-assembly3.cif (C)

*author defined assembly, 1 molecule(s) (monomeric)

7u4r-assembly4.cif.gz Display(72.82 KB)
7u4r-assembly4.cif (D)

*author defined assembly, 1 molecule(s) (monomeric)

7u4r-assembly5.cif.gz Display(71.92 KB)
7u4r-assembly5.cif (E)

*author defined assembly, 1 molecule(s) (monomeric)

7u4r-assembly6.cif.gz Display(72.77 KB)
7u4r-assembly6.cif (F)

*author defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)7u4r.pdb1.gz Display(52.91 KB)
7u4r.pdb1 (A)

*author defined assembly, 1 molecule(s) (monomeric)

7u4r.pdb2.gz Display(52.54 KB)
7u4r.pdb2 (B)

*author defined assembly, 1 molecule(s) (monomeric)

7u4r.pdb3.gz Display(53.06 KB)
7u4r.pdb3 (C)

*author defined assembly, 1 molecule(s) (monomeric)

7u4r.pdb4.gz Display(52.92 KB)
7u4r.pdb4 (D)

*author defined assembly, 1 molecule(s) (monomeric)

7u4r.pdb5.gz Display(52.31 KB)
7u4r.pdb5 (E)

*author defined assembly, 1 molecule(s) (monomeric)

7u4r.pdb6.gz Display(52.78 KB)
7u4r.pdb6 (F)

*author defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF7u4r_validation.pdf.gz Display(1.94 MB)
7u4r_validation.pdf
PDF-full7u4r_full_validation.pdf.gz Display(1.96 MB)
7u4r_full_validation.pdf
mmCIF7u4r_validation.cif.gz Display(42.20 KB)
7u4r_validation.cif
XML7u4r_validation.xml.gz Display(34.68 KB)
7u4r_validation.xml
PNG7u4r_multipercentile_validation.png.gz Display(155.28 KB)
7u4r_multipercentile_validation.png
SVG7u4r_multipercentile_validation.svg.gz Display(950.00 B)
7u4r_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)7u4r_validation_2fo-fc_map_coef.cif.gz Display(241.21 KB)
7u4r_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)7u4r_validation_fo-fc_map_coef.cif.gz Display(213.90 KB)
7u4r_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)7u4r_validation_2fo-fc_map_coef.mtz Visualize(574.09 KB)
fo-fc (MTZ)7u4r_validation_fo-fc_map_coef.mtz Visualize(574.09 KB)

246704

PDB entries from 2025-12-24

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