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6P5P

Discovery of a Novel, Highly Potent, and Selective Thieno[3,2-d]pyrimidinone-Based Cdc7 inhibitor with a Quinuclidine Moiety (TAK-931) as an Orally Active Investigational Anti-Tumor Agent

Resources
File formatFile name (file size)
PDBx/mmCIF6p5p.cif.gz Display(626.45 KB)
6p5p.cif
PDBx/mmJSONall6p5p.json.gz Display (Tree)(405.38 KB)
6p5p.json
no-atom6p5p-noatom.json.gz Display (Header)(21.62 KB)
6p5p-noatom.json
add only6p5p-plus.json.gz Display(1.10 KB)
6p5p-plus.json
PDBMLall6p5p.xml.gz Display(863.99 KB)
6p5p.xml
no-atom6p5p-noatom.xml.gz Display(55.49 KB)
6p5p-noatom.xml
ext-atom6p5p-extatom.xml.gz Display(281.90 KB)
6p5p-extatom.xml
PDBpdb6p5p.ent.gz Display(527.01 KB)
pdb6p5p.ent
RDF6p5p.rdf.gz Visualize(160.23 KB)
6p5p.rdf
Structure factorsr6p5psf.ent.gz Display(1.23 MB)
r6p5psf.ent
Biological unit (mmCIF format)6p5p-assembly1.cif.gz Display(163.20 KB)
6p5p-assembly1.cif (A)

*author defined assembly, 1 molecule(s) (monomeric)

6p5p-assembly2.cif.gz Display(157.60 KB)
6p5p-assembly2.cif (B)

*author defined assembly, 1 molecule(s) (monomeric)

6p5p-assembly3.cif.gz Display(159.04 KB)
6p5p-assembly3.cif (C)

*author defined assembly, 1 molecule(s) (monomeric)

6p5p-assembly4.cif.gz Display(163.20 KB)
6p5p-assembly4.cif (D)

*author defined assembly, 1 molecule(s) (monomeric)

6p5p-assembly5.cif.gz Display(317.96 KB)
6p5p-assembly5.cif (A,D)

*software defined assembly, 2 molecule(s) (dimeric)

6p5p-assembly6.cif.gz Display(308.04 KB)
6p5p-assembly6.cif (B,C)

*software defined assembly, 2 molecule(s) (dimeric)

Biological unit (PDB format)6p5p.pdb1.gz Display(134.23 KB)
6p5p.pdb1 (A)

*author defined assembly, 1 molecule(s) (monomeric)

6p5p.pdb2.gz Display(130.28 KB)
6p5p.pdb2 (B)

*author defined assembly, 1 molecule(s) (monomeric)

6p5p.pdb3.gz Display(132.05 KB)
6p5p.pdb3 (C)

*author defined assembly, 1 molecule(s) (monomeric)

6p5p.pdb4.gz Display(134.98 KB)
6p5p.pdb4 (D)

*author defined assembly, 1 molecule(s) (monomeric)

6p5p.pdb5.gz Display(264.90 KB)
6p5p.pdb5 (A,D)

*software defined assembly, 2 molecule(s) (dimeric)

6p5p.pdb6.gz Display(257.99 KB)
6p5p.pdb6 (B,C)

*software defined assembly, 2 molecule(s) (dimeric)

Validation reportsPDF6p5p_validation.pdf.gz Display(438.90 KB)
6p5p_validation.pdf
PDF-full6p5p_full_validation.pdf.gz Display(441.10 KB)
6p5p_full_validation.pdf
mmCIF6p5p_validation.cif.gz Display(15.35 KB)
6p5p_validation.cif
XML6p5p_validation.xml.gz Display(1.92 KB)
6p5p_validation.xml
EDMap2fo-fc (MTZ)6p5p_validation_2fo-fc_map_coef.mtz Visualize(1016.95 KB)
fo-fc (MTZ)6p5p_validation_fo-fc_map_coef.mtz Visualize(1016.95 KB)

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PDB entries from 2024-07-17

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