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5WHR

Discovery of a novel and selective IDO-1 inhibitor PF-06840003 and its characterization as a potential clinical candidate.

Resources
File formatFile name (file size)
PDBx/mmCIF5whr.cif.gz Display(162.82 KB)
5whr.cif
PDBx/mmJSONall5whr.json.gz Display (Tree)(108.36 KB)
5whr.json
no-atom5whr-noatom.json.gz Display (Header)(16.04 KB)
5whr-noatom.json
add only5whr-plus.json.gz Display(1.71 KB)
5whr-plus.json
PDBMLall5whr.xml.gz Display(219.44 KB)
5whr.xml
no-atom5whr-noatom.xml.gz Display(31.35 KB)
5whr-noatom.xml
ext-atom5whr-extatom.xml.gz Display(140.72 KB)
5whr-extatom.xml
PDBpdb5whr.ent.gz Display(133.58 KB)
pdb5whr.ent
RDF5whr.rdf.gz Visualize(80.48 KB)
5whr.rdf
Structure factorsr5whrsf.ent.gz Display(1.56 MB)
r5whrsf.ent
Biological unit (mmCIF format)5whr-assembly1.cif.gz Display(156.15 KB)
5whr-assembly1.cif (A,B)

*author defined assembly, 2 molecule(s) (dimeric)

Biological unit (PDB format)5whr.pdb1.gz Display(128.12 KB)
5whr.pdb1 (A,B)

*author defined assembly, 2 molecule(s) (dimeric)

Validation reportsPDF5whr_validation.pdf.gz Display(1.77 MB)
5whr_validation.pdf
PDF-full5whr_full_validation.pdf.gz Display(1.78 MB)
5whr_full_validation.pdf
mmCIF5whr_validation.cif.gz Display(43.15 KB)
5whr_validation.cif
XML5whr_validation.xml.gz Display(30.51 KB)
5whr_validation.xml
PNG5whr_multipercentile_validation.png.gz Display(170.00 KB)
5whr_multipercentile_validation.png
SVG5whr_multipercentile_validation.svg.gz Display(975.00 B)
5whr_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)5whr_validation_2fo-fc_map_coef.cif.gz Display(697.56 KB)
5whr_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)5whr_validation_fo-fc_map_coef.cif.gz Display(698.65 KB)
5whr_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)5whr_validation_2fo-fc_map_coef.mtz Visualize(1.09 MB)
fo-fc (MTZ)5whr_validation_fo-fc_map_coef.mtz Visualize(1.09 MB)

224004

PDB entries from 2024-08-21

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