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5WEV

Identification of an imidazopyridine scaffold to generate potent and selective TYK2 inhibitors that demonstrate activity in an in vivo psoriasis model

Resources
File formatFile name (file size)
PDBx/mmCIF5wev.cif.gz Display(82.20 KB)
5wev.cif
PDBx/mmJSONall5wev.json.gz Display (Tree)(58.13 KB)
5wev.json
no-atom5wev-noatom.json.gz Display (Header)(16.17 KB)
5wev-noatom.json
add only5wev-plus.json.gz Display(1.17 KB)
5wev-plus.json
PDBMLall5wev.xml.gz Display(105.67 KB)
5wev.xml
no-atom5wev-noatom.xml.gz Display(26.37 KB)
5wev-noatom.xml
ext-atom5wev-extatom.xml.gz Display(59.27 KB)
5wev-extatom.xml
PDBpdb5wev.ent.gz Display(58.27 KB)
pdb5wev.ent
RDF5wev.rdf.gz Visualize(78.41 KB)
5wev.rdf
Structure factorsr5wevsf.ent.gz Display(888.91 KB)
r5wevsf.ent
Biological unit (mmCIF format)5wev-assembly1.cif.gz Display(69.86 KB)
5wev-assembly1.cif (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)5wev.pdb1.gz Display(53.44 KB)
5wev.pdb1 (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF5wev_validation.pdf.gz Display(781.67 KB)
5wev_validation.pdf
PDF-full5wev_full_validation.pdf.gz Display(783.95 KB)
5wev_full_validation.pdf
mmCIF5wev_validation.cif.gz Display(20.11 KB)
5wev_validation.cif
XML5wev_validation.xml.gz Display(14.45 KB)
5wev_validation.xml
PNG5wev_multipercentile_validation.png.gz Display(158.65 KB)
5wev_multipercentile_validation.png
SVG5wev_multipercentile_validation.svg.gz Display(919.00 B)
5wev_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)5wev_validation_2fo-fc_map_coef.cif.gz Display(311.82 KB)
5wev_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)5wev_validation_fo-fc_map_coef.cif.gz Display(301.17 KB)
5wev_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)5wev_validation_2fo-fc_map_coef.mtz Visualize(738.73 KB)
fo-fc (MTZ)5wev_validation_fo-fc_map_coef.mtz Visualize(738.73 KB)

223166

PDB entries from 2024-07-31

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