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5TO8

Selectivity switch between FAK and Pyk2: Macrocyclization of FAK inhibitors improves Pyk2 potency

Resources
File formatFile name (file size)
PDBx/mmCIF5to8.cif.gz Display(66.81 KB)
5to8.cif
PDBx/mmJSONall5to8.json.gz Display (Tree)(47.22 KB)
5to8.json
no-atom5to8-noatom.json.gz Display (Header)(14.43 KB)
5to8-noatom.json
add only5to8-plus.json.gz Display(1.24 KB)
5to8-plus.json
PDBMLall5to8.xml.gz Display(87.57 KB)
5to8.xml
no-atom5to8-noatom.xml.gz Display(25.05 KB)
5to8-noatom.xml
ext-atom5to8-extatom.xml.gz Display(46.79 KB)
5to8-extatom.xml
pdb_nextgenallpdb_00005to8_xyz-enrich.cif.gz Display(75.19 KB)
pdb_00005to8_xyz-enrich.cif
no-atompdb_00005to8_xyz-no-atom-enrich.xml.gz Display(35.57 KB)
pdb_00005to8_xyz-no-atom-enrich.xml
ng-only5to8-plus.json.gz Display(2.76 KB)
5to8-plus.json
PDBpdb5to8.ent.gz Display(46.99 KB)
pdb5to8.ent
RDF5to8.rdf.gz Visualize(75.05 KB)
5to8.rdf
Structure factorsr5to8sf.ent.gz Display(314.37 KB)
r5to8sf.ent
Biological unit (mmCIF format)5to8-assembly1.cif.gz Display(55.35 KB)
5to8-assembly1.cif (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)5to8.pdb1.gz Display(42.35 KB)
5to8.pdb1 (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF5to8_validation.pdf.gz Display(829.32 KB)
5to8_validation.pdf
PDF-full5to8_full_validation.pdf.gz Display(830.95 KB)
5to8_full_validation.pdf
mmCIF5to8_validation.cif.gz Display(16.63 KB)
5to8_validation.cif
XML5to8_validation.xml.gz Display(12.27 KB)
5to8_validation.xml
PNG5to8_multipercentile_validation.png.gz Display(169.91 KB)
5to8_multipercentile_validation.png
SVG5to8_multipercentile_validation.svg.gz Display(957.00 B)
5to8_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)5to8_validation_2fo-fc_map_coef.cif.gz Display(302.00 KB)
5to8_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)5to8_validation_fo-fc_map_coef.cif.gz Display(295.18 KB)
5to8_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)5to8_validation_2fo-fc_map_coef.mtz Visualize(486.16 KB)
fo-fc (MTZ)5to8_validation_fo-fc_map_coef.mtz Visualize(486.16 KB)

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PDB entries from 2026-01-14

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