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5SIO

CRYSTAL STRUCTURE OF HUMAN PHOSPHODIESTERASE 10 IN COMPLEX WITH C(=O)(N1CCCC1C)c5c(C(Nc3cc2nc(cn2cc3)c4ccccc4)=O)n(nc5)C, micromolar IC50=0.000107

Resources
File formatFile name (file size)
PDBx/mmCIF5sio.cif.gz Display(274.83 KB)
5sio.cif
PDBx/mmJSONall5sio.json.gz Display (Tree)(169.77 KB)
5sio.json
no-atom5sio-noatom.json.gz Display (Header)(20.97 KB)
5sio-noatom.json
add only5sio-plus.json.gz Display(1.02 KB)
5sio-plus.json
PDBMLall5sio.xml.gz Display(376.16 KB)
5sio.xml
no-atom5sio-noatom.xml.gz Display(56.24 KB)
5sio-noatom.xml
ext-atom5sio-extatom.xml.gz Display(242.03 KB)
5sio-extatom.xml
pdb_nextgenallpdb_00005sio_xyz-enrich.cif.gz Display(299.98 KB)
pdb_00005sio_xyz-enrich.cif
no-atompdb_00005sio_xyz-no-atom-enrich.xml.gz Display(68.93 KB)
pdb_00005sio_xyz-no-atom-enrich.xml
ng-only5sio-plus.json.gz Display(3.41 KB)
5sio-plus.json
PDBpdb5sio.ent.gz Display(221.39 KB)
pdb5sio.ent
RDF5sio.rdf.gz Visualize(152.18 KB)
5sio.rdf
Structure factorsr5siosf.ent.gz Display(8.84 MB)
r5siosf.ent
Biological unit (mmCIF format)5sio-assembly1.cif.gz Display(71.57 KB)
5sio-assembly1.cif (A)

*author defined assembly, 1 molecule(s) (monomeric)

5sio-assembly2.cif.gz Display(71.76 KB)
5sio-assembly2.cif (B)

*author defined assembly, 1 molecule(s) (monomeric)

5sio-assembly3.cif.gz Display(71.30 KB)
5sio-assembly3.cif (C)

*author defined assembly, 1 molecule(s) (monomeric)

5sio-assembly4.cif.gz Display(69.16 KB)
5sio-assembly4.cif (D)

*author defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)5sio.pdb1.gz Display(56.85 KB)
5sio.pdb1 (A)

*author defined assembly, 1 molecule(s) (monomeric)

5sio.pdb2.gz Display(57.04 KB)
5sio.pdb2 (B)

*author defined assembly, 1 molecule(s) (monomeric)

5sio.pdb3.gz Display(56.79 KB)
5sio.pdb3 (C)

*author defined assembly, 1 molecule(s) (monomeric)

5sio.pdb4.gz Display(55.34 KB)
5sio.pdb4 (D)

*author defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF5sio_validation.pdf.gz Display(1.31 MB)
5sio_validation.pdf
PDF-full5sio_full_validation.pdf.gz Display(1.32 MB)
5sio_full_validation.pdf
mmCIF5sio_validation.cif.gz Display(74.41 KB)
5sio_validation.cif
XML5sio_validation.xml.gz Display(57.38 KB)
5sio_validation.xml
PNG5sio_multipercentile_validation.png.gz Display(173.92 KB)
5sio_multipercentile_validation.png
SVG5sio_multipercentile_validation.svg.gz Display(976.00 B)
5sio_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)5sio_validation_2fo-fc_map_coef.cif.gz Display(1.20 MB)
5sio_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)5sio_validation_fo-fc_map_coef.cif.gz Display(1.18 MB)
5sio_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)5sio_validation_2fo-fc_map_coef.mtz Visualize(1.87 MB)
fo-fc (MTZ)5sio_validation_fo-fc_map_coef.mtz Visualize(1.87 MB)

238895

PDB entries from 2025-07-16

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