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5SI0

CRYSTAL STRUCTURE OF HUMAN PHOSPHODIESTERASE 10 IN COMPLEX WITH n4c(n1c(nc(n1)CCc2nn(c(n2)N3CCCC3)C)cc4C)CCc5nn(c(n5)N6CCCC6)C, micromolar IC50=0.047938

Resources
File formatFile name (file size)
PDBx/mmCIF5si0.cif.gz Display(269.67 KB)
5si0.cif
PDBx/mmJSONall5si0.json.gz Display (Tree)(167.91 KB)
5si0.json
no-atom5si0-noatom.json.gz Display (Header)(19.48 KB)
5si0-noatom.json
add only5si0-plus.json.gz Display(1011.00 B)
5si0-plus.json
PDBMLall5si0.xml.gz Display(370.78 KB)
5si0.xml
no-atom5si0-noatom.xml.gz Display(53.34 KB)
5si0-noatom.xml
ext-atom5si0-extatom.xml.gz Display(239.44 KB)
5si0-extatom.xml
pdb_nextgenallpdb_00005si0_xyz-enrich.cif.gz Display(294.55 KB)
pdb_00005si0_xyz-enrich.cif
no-atompdb_00005si0_xyz-no-atom-enrich.xml.gz Display(66.49 KB)
pdb_00005si0_xyz-no-atom-enrich.xml
ng-only5si0-plus.json.gz Display(3.42 KB)
5si0-plus.json
PDBpdb5si0.ent.gz Display(218.82 KB)
pdb5si0.ent
RDF5si0.rdf.gz Visualize(147.64 KB)
5si0.rdf
Structure factorsr5si0sf.ent.gz Display(8.95 MB)
r5si0sf.ent
Biological unit (mmCIF format)5si0-assembly1.cif.gz Display(70.72 KB)
5si0-assembly1.cif (A)

*author defined assembly, 1 molecule(s) (monomeric)

5si0-assembly2.cif.gz Display(69.95 KB)
5si0-assembly2.cif (B)

*author defined assembly, 1 molecule(s) (monomeric)

5si0-assembly3.cif.gz Display(69.69 KB)
5si0-assembly3.cif (C)

*author defined assembly, 1 molecule(s) (monomeric)

5si0-assembly4.cif.gz Display(67.54 KB)
5si0-assembly4.cif (D)

*author defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)5si0.pdb1.gz Display(56.81 KB)
5si0.pdb1 (A)

*author defined assembly, 1 molecule(s) (monomeric)

5si0.pdb2.gz Display(56.05 KB)
5si0.pdb2 (B)

*author defined assembly, 1 molecule(s) (monomeric)

5si0.pdb3.gz Display(55.88 KB)
5si0.pdb3 (C)

*author defined assembly, 1 molecule(s) (monomeric)

5si0.pdb4.gz Display(54.03 KB)
5si0.pdb4 (D)

*author defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF5si0_validation.pdf.gz Display(1.66 MB)
5si0_validation.pdf
PDF-full5si0_full_validation.pdf.gz Display(1.68 MB)
5si0_full_validation.pdf
mmCIF5si0_validation.cif.gz Display(71.22 KB)
5si0_validation.cif
XML5si0_validation.xml.gz Display(55.30 KB)
5si0_validation.xml
PNG5si0_multipercentile_validation.png.gz Display(170.48 KB)
5si0_multipercentile_validation.png
SVG5si0_multipercentile_validation.svg.gz Display(974.00 B)
5si0_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)5si0_validation_2fo-fc_map_coef.cif.gz Display(1.07 MB)
5si0_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)5si0_validation_fo-fc_map_coef.cif.gz Display(1.08 MB)
5si0_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)5si0_validation_2fo-fc_map_coef.mtz Visualize(1.70 MB)
fo-fc (MTZ)5si0_validation_fo-fc_map_coef.mtz Visualize(1.70 MB)

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PDB entries from 2026-01-14

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