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5SHR

CRYSTAL STRUCTURE OF HUMAN PHOSPHODIESTERASE 10 IN COMPLEX WITH n1(c(nc(n1)c2ccccc2)N(C)Cc4nn3c(cnc(c3n4)C)C)C, micromolar IC50=1.47052

Resources
File formatFile name (file size)
PDBx/mmCIF5shr.cif.gz Display(276.22 KB)
5shr.cif
PDBx/mmJSONall5shr.json.gz Display (Tree)(169.98 KB)
5shr.json
no-atom5shr-noatom.json.gz Display (Header)(20.71 KB)
5shr-noatom.json
add only5shr-plus.json.gz Display(1.05 KB)
5shr-plus.json
PDBMLall5shr.xml.gz Display(378.22 KB)
5shr.xml
no-atom5shr-noatom.xml.gz Display(57.13 KB)
5shr-noatom.xml
ext-atom5shr-extatom.xml.gz Display(242.87 KB)
5shr-extatom.xml
pdb_nextgenallpdb_00005shr_xyz-enrich.cif.gz Display(302.34 KB)
pdb_00005shr_xyz-enrich.cif
no-atompdb_00005shr_xyz-no-atom-enrich.xml.gz Display(70.33 KB)
pdb_00005shr_xyz-no-atom-enrich.xml
ng-only5shr-plus.json.gz Display(3.43 KB)
5shr-plus.json
PDBpdb5shr.ent.gz Display(221.72 KB)
pdb5shr.ent
RDF5shr.rdf.gz Visualize(160.19 KB)
5shr.rdf
Structure factorsr5shrsf.ent.gz Display(13.36 MB)
r5shrsf.ent
Biological unit (mmCIF format)5shr-assembly1.cif.gz Display(71.37 KB)
5shr-assembly1.cif (A)

*author defined assembly, 1 molecule(s) (monomeric)

5shr-assembly2.cif.gz Display(71.88 KB)
5shr-assembly2.cif (B)

*author defined assembly, 1 molecule(s) (monomeric)

5shr-assembly3.cif.gz Display(71.65 KB)
5shr-assembly3.cif (C)

*author defined assembly, 1 molecule(s) (monomeric)

5shr-assembly4.cif.gz Display(69.53 KB)
5shr-assembly4.cif (D)

*author defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)5shr.pdb1.gz Display(56.61 KB)
5shr.pdb1 (A)

*author defined assembly, 1 molecule(s) (monomeric)

5shr.pdb2.gz Display(56.99 KB)
5shr.pdb2 (B)

*author defined assembly, 1 molecule(s) (monomeric)

5shr.pdb3.gz Display(56.87 KB)
5shr.pdb3 (C)

*author defined assembly, 1 molecule(s) (monomeric)

5shr.pdb4.gz Display(55.25 KB)
5shr.pdb4 (D)

*author defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF5shr_validation.pdf.gz Display(1.49 MB)
5shr_validation.pdf
PDF-full5shr_full_validation.pdf.gz Display(1.51 MB)
5shr_full_validation.pdf
mmCIF5shr_validation.cif.gz Display(77.13 KB)
5shr_validation.cif
XML5shr_validation.xml.gz Display(59.17 KB)
5shr_validation.xml
PNG5shr_multipercentile_validation.png.gz Display(170.47 KB)
5shr_multipercentile_validation.png
SVG5shr_multipercentile_validation.svg.gz Display(975.00 B)
5shr_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)5shr_validation_2fo-fc_map_coef.cif.gz Display(1.53 MB)
5shr_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)5shr_validation_fo-fc_map_coef.cif.gz Display(1.53 MB)
5shr_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)5shr_validation_2fo-fc_map_coef.mtz Visualize(2.55 MB)
fo-fc (MTZ)5shr_validation_fo-fc_map_coef.mtz Visualize(2.55 MB)

247536

PDB entries from 2026-01-14

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