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5IU2

Discovery of imidazoquinolines as a novel class of potent, selective and in vivo efficacious COT kinase inhibitors

Replaces:  4Y83Replaces:  4Y85
Resources
File formatFile name (file size)
PDBx/mmCIF5iu2.cif.gz Display(251.45 KB)
5iu2.cif
PDBx/mmJSONall5iu2.json.gz Display (Tree)(169.26 KB)
5iu2.json
no-atom5iu2-noatom.json.gz Display (Header)(17.22 KB)
5iu2-noatom.json
add only5iu2-plus.json.gz Display(1.21 KB)
5iu2-plus.json
PDBMLall5iu2.xml.gz Display(346.93 KB)
5iu2.xml
no-atom5iu2-noatom.xml.gz Display(36.03 KB)
5iu2-noatom.xml
ext-atom5iu2-extatom.xml.gz Display(112.27 KB)
5iu2-extatom.xml
PDBpdb5iu2.ent.gz Display(201.03 KB)
pdb5iu2.ent
RDF5iu2.rdf.gz Visualize(105.45 KB)
5iu2.rdf
Structure factorsr5iu2sf.ent.gz Display(244.76 KB)
r5iu2sf.ent
Biological unit (mmCIF format)5iu2-assembly1.cif.gz Display(124.83 KB)
5iu2-assembly1.cif (A)

*author defined assembly, 1 molecule(s) (monomeric)

5iu2-assembly2.cif.gz Display(124.16 KB)
5iu2-assembly2.cif (B)

*author defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)5iu2.pdb1.gz Display(99.21 KB)
5iu2.pdb1 (A)

*author defined assembly, 1 molecule(s) (monomeric)

5iu2.pdb2.gz Display(99.13 KB)
5iu2.pdb2 (B)

*author defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF5iu2_validation.pdf.gz Display(1008.04 KB)
5iu2_validation.pdf
PDF-full5iu2_full_validation.pdf.gz Display(1010.66 KB)
5iu2_full_validation.pdf
mmCIF5iu2_validation.cif.gz Display(34.66 KB)
5iu2_validation.cif
XML5iu2_validation.xml.gz Display(24.82 KB)
5iu2_validation.xml
PNG5iu2_multipercentile_validation.png.gz Display(173.68 KB)
5iu2_multipercentile_validation.png
SVG5iu2_multipercentile_validation.svg.gz Display(979.00 B)
5iu2_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)5iu2_validation_2fo-fc_map_coef.cif.gz Display(202.88 KB)
5iu2_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)5iu2_validation_fo-fc_map_coef.cif.gz Display(198.88 KB)
5iu2_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)5iu2_validation_2fo-fc_map_coef.mtz Visualize(481.32 KB)
fo-fc (MTZ)5iu2_validation_fo-fc_map_coef.mtz Visualize(481.32 KB)

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PDB entries from 2024-07-10

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