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4V25

VER-246608, a novel pan-isoform ATP competitive inhibitor of pyruvate dehydrogenase kinase, disrupts Warburg metabolism and induces context- dependent cytostasis in cancer cells

Resources
File formatFile name (file size)
PDBx/mmCIF4v25.cif.gz Display(87.20 KB)
4v25.cif
PDBx/mmJSONall4v25.json.gz Display (Tree)(60.71 KB)
4v25.json
no-atom4v25-noatom.json.gz Display (Header)(14.75 KB)
4v25-noatom.json
add only4v25-plus.json.gz Display(1.36 KB)
4v25-plus.json
PDBMLall4v25.xml.gz Display(116.78 KB)
4v25.xml
no-atom4v25-noatom.xml.gz Display(29.24 KB)
4v25-noatom.xml
ext-atom4v25-extatom.xml.gz Display(65.95 KB)
4v25-extatom.xml
PDBpdb4v25.ent.gz Display(65.56 KB)
pdb4v25.ent
RDF4v25.rdf.gz Visualize(89.71 KB)
4v25.rdf
Structure factorsr4v25sf.ent.gz Display(326.55 KB)
r4v25sf.ent
Biological unit (mmCIF format)4v25-assembly1.cif.gz Display(145.37 KB)
4v25-assembly1.cif (A)

*author and software defined assembly, 2 molecule(s) (dimeric)

Biological unit (PDB format)4v25.pdb1.gz Display(116.05 KB)
4v25.pdb1 (A)

*author and software defined assembly, 2 molecule(s) (dimeric)

Validation reportsPDF4v25_validation.pdf.gz Display(937.93 KB)
4v25_validation.pdf
PDF-full4v25_full_validation.pdf.gz Display(944.22 KB)
4v25_full_validation.pdf
mmCIF4v25_validation.cif.gz Display(21.74 KB)
4v25_validation.cif
XML4v25_validation.xml.gz Display(15.91 KB)
4v25_validation.xml
PNG4v25_multipercentile_validation.png.gz Display(165.68 KB)
4v25_multipercentile_validation.png
SVG4v25_multipercentile_validation.svg.gz Display(979.00 B)
4v25_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)4v25_validation_2fo-fc_map_coef.cif.gz Display(262.79 KB)
4v25_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)4v25_validation_fo-fc_map_coef.cif.gz Display(259.29 KB)
4v25_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)4v25_validation_2fo-fc_map_coef.mtz Visualize(415.55 KB)
fo-fc (MTZ)4v25_validation_fo-fc_map_coef.mtz Visualize(415.55 KB)

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PDB entries from 2024-07-24

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