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4P7E

Triazolopyridine compounds as selective JAK1 inhibitors: from hit identification to GLPG0634

Resources
File formatFile name (file size)
PDBx/mmCIF4p7e.cif.gz Display(137.17 KB)
4p7e.cif
PDBx/mmJSONall4p7e.json.gz Display (Tree)(90.40 KB)
4p7e.json
no-atom4p7e-noatom.json.gz Display (Header)(16.58 KB)
4p7e-noatom.json
add only4p7e-plus.json.gz Display(1.23 KB)
4p7e-plus.json
PDBMLall4p7e.xml.gz Display(184.95 KB)
4p7e.xml
no-atom4p7e-noatom.xml.gz Display(35.11 KB)
4p7e-noatom.xml
ext-atom4p7e-extatom.xml.gz Display(113.31 KB)
4p7e-extatom.xml
pdb_nextgenallpdb_00004p7e_xyz-enrich.cif.gz Display(155.06 KB)
pdb_00004p7e_xyz-enrich.cif
no-atompdb_00004p7e_xyz-no-atom-enrich.xml.gz Display(56.20 KB)
pdb_00004p7e_xyz-no-atom-enrich.xml
ng-only4p7e-plus.json.gz Display(3.57 KB)
4p7e-plus.json
PDBpdb4p7e.ent.gz Display(106.26 KB)
pdb4p7e.ent
RDF4p7e.rdf.gz Visualize(97.51 KB)
4p7e.rdf
Structure factorsr4p7esf.ent.gz Display(1.98 MB)
r4p7esf.ent
Biological unit (mmCIF format)4p7e-assembly1.cif.gz Display(66.85 KB)
4p7e-assembly1.cif (A)

*software defined assembly, 1 molecule(s) (monomeric)

4p7e-assembly2.cif.gz Display(67.00 KB)
4p7e-assembly2.cif (B)

*software defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)4p7e.pdb1.gz Display(52.03 KB)
4p7e.pdb1 (A)

*software defined assembly, 1 molecule(s) (monomeric)

4p7e.pdb2.gz Display(51.82 KB)
4p7e.pdb2 (B)

*software defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF4p7e_validation.pdf.gz Display(1016.60 KB)
4p7e_validation.pdf
PDF-full4p7e_full_validation.pdf.gz Display(1.00 MB)
4p7e_full_validation.pdf
mmCIF4p7e_validation.cif.gz Display(36.54 KB)
4p7e_validation.cif
XML4p7e_validation.xml.gz Display(26.53 KB)
4p7e_validation.xml
PNG4p7e_multipercentile_validation.png.gz Display(172.08 KB)
4p7e_multipercentile_validation.png
SVG4p7e_multipercentile_validation.svg.gz Display(957.00 B)
4p7e_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)4p7e_validation_2fo-fc_map_coef.cif.gz Display(342.82 KB)
4p7e_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)4p7e_validation_fo-fc_map_coef.cif.gz Display(335.61 KB)
4p7e_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)4p7e_validation_2fo-fc_map_coef.mtz Visualize(805.98 KB)
fo-fc (MTZ)4p7e_validation_fo-fc_map_coef.mtz Visualize(805.98 KB)

246704

PDB entries from 2025-12-24

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