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4I11

Structure-based design of novel dihydroisoquinoline BACE-1 inhibitors that do not engage the catalytic aspartates.

Resources
File formatFile name (file size)
PDBx/mmCIF4i11.cif.gz Display(97.41 KB)
4i11.cif
PDBx/mmJSONall4i11.json.gz Display (Tree)(69.27 KB)
4i11.json
no-atom4i11-noatom.json.gz Display (Header)(15.24 KB)
4i11-noatom.json
add only4i11-plus.json.gz Display(1.10 KB)
4i11-plus.json
PDBMLall4i11.xml.gz Display(130.12 KB)
4i11.xml
no-atom4i11-noatom.xml.gz Display(26.44 KB)
4i11-noatom.xml
ext-atom4i11-extatom.xml.gz Display(78.26 KB)
4i11-extatom.xml
PDBpdb4i11.ent.gz Display(77.70 KB)
pdb4i11.ent
RDF4i11.rdf.gz Visualize(63.52 KB)
4i11.rdf
Structure factorsr4i11sf.ent.gz Display(455.40 KB)
r4i11sf.ent
Biological unit (mmCIF format)4i11-assembly1.cif.gz Display(91.17 KB)
4i11-assembly1.cif (A)

*author defined assembly, 1 molecule(s) (monomeric)

4i11-assembly2.cif.gz Display(173.25 KB)
4i11-assembly2.cif (A)

*software defined assembly, 2 molecule(s) (dimeric)

Biological unit (PDB format)4i11.pdb1.gz Display(71.94 KB)
4i11.pdb1 (A)

*author defined assembly, 1 molecule(s) (monomeric)

4i11.pdb2.gz Display(140.82 KB)
4i11.pdb2 (A)

*software defined assembly, 2 molecule(s) (dimeric)

Validation reportsPDF4i11_validation.pdf.gz Display(812.10 KB)
4i11_validation.pdf
PDF-full4i11_full_validation.pdf.gz Display(816.75 KB)
4i11_full_validation.pdf
mmCIF4i11_validation.cif.gz Display(29.80 KB)
4i11_validation.cif
XML4i11_validation.xml.gz Display(19.77 KB)
4i11_validation.xml
PNG4i11_multipercentile_validation.png.gz Display(168.31 KB)
4i11_multipercentile_validation.png
SVG4i11_multipercentile_validation.svg.gz Display(960.00 B)
4i11_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)4i11_validation_2fo-fc_map_coef.cif.gz Display(463.31 KB)
4i11_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)4i11_validation_fo-fc_map_coef.cif.gz Display(444.43 KB)
4i11_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)4i11_validation_2fo-fc_map_coef.mtz Visualize(753.30 KB)
fo-fc (MTZ)4i11_validation_fo-fc_map_coef.mtz Visualize(753.30 KB)

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PDB entries from 2024-07-17

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