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3KL6

Discovery of Tetrahydropyrimidin-2(1H)-one derivative TAK-442: A potent, selective and orally active factor Xa inhibitor

Resources
File formatFile name (file size)
PDBx/mmCIF3kl6.cif.gz Display(77.66 KB)
3kl6.cif
PDBx/mmJSONall3kl6.json.gz Display (Tree)(54.71 KB)
3kl6.json
no-atom3kl6-noatom.json.gz Display (Header)(15.63 KB)
3kl6-noatom.json
add only3kl6-plus.json.gz Display(1.24 KB)
3kl6-plus.json
PDBMLall3kl6.xml.gz Display(103.05 KB)
3kl6.xml
no-atom3kl6-noatom.xml.gz Display(29.70 KB)
3kl6-noatom.xml
ext-atom3kl6-extatom.xml.gz Display(54.46 KB)
3kl6-extatom.xml
PDBpdb3kl6.ent.gz Display(55.00 KB)
pdb3kl6.ent
RDF3kl6.rdf.gz Visualize(83.53 KB)
3kl6.rdf
Structure factorsr3kl6sf.ent.gz Display(688.88 KB)
r3kl6sf.ent
Biological unit (mmCIF format)3kl6-assembly1.cif.gz Display(65.26 KB)
3kl6-assembly1.cif (A,B)

*author and software defined assembly, 2 molecule(s) (dimeric)

Biological unit (PDB format)3kl6.pdb1.gz Display(49.70 KB)
3kl6.pdb1 (A,B)

*author and software defined assembly, 2 molecule(s) (dimeric)

Validation reportsPDF3kl6_validation.pdf.gz Display(766.24 KB)
3kl6_validation.pdf
PDF-full3kl6_full_validation.pdf.gz Display(767.74 KB)
3kl6_full_validation.pdf
mmCIF3kl6_validation.cif.gz Display(20.98 KB)
3kl6_validation.cif
XML3kl6_validation.xml.gz Display(14.80 KB)
3kl6_validation.xml
PNG3kl6_multipercentile_validation.png.gz Display(163.20 KB)
3kl6_multipercentile_validation.png
SVG3kl6_multipercentile_validation.svg.gz Display(957.00 B)
3kl6_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)3kl6_validation_2fo-fc_map_coef.cif.gz Display(469.59 KB)
3kl6_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)3kl6_validation_fo-fc_map_coef.cif.gz Display(453.94 KB)
3kl6_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)3kl6_validation_2fo-fc_map_coef.mtz Visualize(1.11 MB)
fo-fc (MTZ)3kl6_validation_fo-fc_map_coef.mtz Visualize(1.11 MB)

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PDB entries from 2024-08-07

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